日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of SD-965 as a Potent, Selective, and Efficacious STAT3 PROTAC Degrader

发现 SD-965 是一种高效、选择性强且有效的 STAT3 PROTAC 降解剂

Wu, Dimin; Zhou, Haibin; Bai, Longchuan; Acharyya, Ranjan Kumar; Metwally, Hoda; McEachern, Donna; Wang, Mi; Tošović, Jelena; Rej, Rohan Kalyan; Wang, Meilin; Wen, Bo; Sun, Duxin; Wang, Shaomeng

circOMA1 delivered by exosomes regulates DRD2‑mediated prolactinoma resistance.

外泌体递送的 circOMA1 调节 DRD2 介导的催乳素瘤耐药性。

Rao Qing, Zhu Dimin, Wang Zongming, Zhang Shaolin, Li Xueli, Tagilapalli Shashikiran, Wang Nan, Hu Weiyu, Chen Wenli, Zhu Yonghong

Serum starvation-induced cholesterol reduction increases melanoma cell susceptibility to cytotoxic T lymphocyte killing

血清饥饿诱导的胆固醇降低会增加黑色素瘤细胞对细胞毒性T淋巴细胞杀伤的敏感性

Miaomiao Hou,Longtao Ji,Dimin Li,Qian Xiao,Xiao Hu

Pediatric pancreatic acinar cell carcinoma with a non-canonical BRAF-KMT2C fusion and a classic SND1-BRAF fusion: a case report and literature review

儿童胰腺腺泡细胞癌伴非典型BRAF-KMT2C融合和经典SND1-BRAF融合:病例报告及文献综述

Wang, Yaqin; Zhang, Jiasi; Nie, Dimin; Zhang, Ai; Hu, Qun; Liu, Aiguo

Discovery of ERD-1233 as a Potent and Orally Efficacious Estrogen Receptor PROTAC Degrader for the Treatment of ER+ Human Breast Cancer

发现 ERD-1233 是一种强效且口服有效的雌激素受体 PROTAC 降解剂,可用于治疗 ER+ 人类乳腺癌

Acharyya, Ranjan Kumar; Rej, Rohan Kalyan; Hu, Biao; Chen, Zhixiang; Wu, Dimin; Lu, Jianfeng; Metwally, Hoda; McEachern, Donna; Wang, Yu; Jiang, Wei; Bai, Longchuan; Tošović, Jelena; Gersch, Christina L; Xu, Guozhang; Zhang, Weihong; Wu, WenXue; Priestley, E Scott; Sui, Zhihua; Sarkari, Farzad; Wen, Bo; Sun, Duxin; Rae, James M; Wang, Shaomeng

Discovery of SD-436: A Potent, Highly Selective and Efficacious STAT3 PROTAC Degrader Capable of Achieving Complete and Long-Lasting Tumor Regression

SD-436 的发现:一种强效、高选择性和高效的 STAT3 PROTAC 降解剂,能够实现完全且持久的肿瘤消退

Xu, Renqi; Zhou, Haibin; Bai, Longchuan; McEachern, Donna; Wu, Dimin; Acharyya, Ranjan Kumar; Wang, Mi; Tošović, Jelena; Yang, Chao-Yie; Chinnaswamy, Krishnapriya; Meagher, Jennifer L; Stuckey, Jeanne A; Liu, Cai; Wang, Meilin; Wen, Bo; Sun, Duxin; Wang, Shaomeng

Discovery of ERD-12310A as an Exceptionally Potent and Orally Efficacious PROTAC Degrader of Estrogen Receptor α (ERα).

发现 ERD-12310A 是一种效力极强且口服有效的雌激素受体 α (ERα) PROTAC 降解剂。

Rej Rohan Kalyan, Hu Biao, Chen Zhixiang, Acharyya Ranjan Kumar, Wu Dimin, Metwally Hoda, McEachern Donna, Wang Yu, Jiang Wei, Bai Longchuan, Nishimura Leticia S, Gersch Christina L, Wang Meilin, Wen Bo, Sun Duxin, Carlson Kathryn, Katzenellenbogen John A, Xu Guozhang, Zhang Weihong, Wu Wenxue, Priestley E Scott, Sui Zhihua, Rae James M, Wang Shaomeng

mTORC1 accelerates osteosarcoma progression via m6A-dependent stabilization of USP7 mRNA

mTORC1 通过 m6A 依赖的 USP7 mRNA 稳定来加速骨肉瘤进展

Zhengming Yang #, Wei Yu #, Ankai Xu, Bing Liu, Libin Jin, Huimin Tao, Dimin Wang

Clinical application of combination [(11)C]C-methionine and [(13)N]N-ammonia PET/CT in recurrent functional pituitary adenomas with negative MRI or [(18)F]F-FDG PET/CT

[(11)C]C-蛋氨酸和[(13)N]N-氨PET/CT联合应用在MRI或[(18)F]F-FDG PET/CT阴性的复发性功能性垂体腺瘤中的临床应用

Wang, Zongming; Feng, Zize; Zhu, Dimin; Wang, Xin; Chen, Jinping; Zhu, Yonghong; Wang, Haijun

Dietary potassium stimulates Ppp1Ca-Ppp1r1a dephosphorylation of kidney NaCl cotransporter and reduces blood pressure

膳食钾可刺激肾脏钠氯共转运蛋白Ppp1Ca-Ppp1r1a去磷酸化,从而降低血压。

Grimm, P Richard; Tatomir, Anamaria; Rosenbaek, Lena L; Kim, Bo Young; Li, Dimin; Delpire, Eric J; Fenton, Robert A; Welling, Paul A