日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Insights from aquaporin structures into drug-resistant sleeping sickness

从水通道蛋白结构中揭示耐药性昏睡病的机制

Matusevicius, Modestas; Corey, Robin A; Gragera, Marcos; Yamashita, Keitaro; Sprenger, Teresa; Ungogo, Marzuq; Blaza, James N; Castro-Hartmann, Pablo; Chirgadze, Dimitri Y; Chaitanya Vedithi, Sundeep; Afanasyev, Pavel; Melero, Roberto; Warshamanage, Rangana; Gusach, Anastasiia; Carazo, José-Maria; Carrington, Mark; Blundell, Tom; Murshudov, Garib N; Stansfeld, Phillip J; Sansom, Mark S P; De Koning, Harry P; Tate, Christopher G; Weyand, Simone

Cryo-EM structures of NHEJ assemblies with nucleosomes

核小体参与的NHEJ组装体的冷冻电镜结构

Hall, Chloe; Frit, Philippe; Kefala-Stavridi, Antonia; Pelletier, Amandine; Hardwick, Steven W; Amin, Himani; Bilyard, Matthew K; Maia De Oliviera, Taiana; Tariq, Ammarah; Zahid, Sayma; Chirgadze, Dimitri Y; Balasubramanian, Shankar; Meek, Katheryn; Ropars, Virginie; Charbonnier, Jean-Baptiste; Modesti, Mauro; Calsou, Patrick; Britton, Sébastien; Blundell, Tom L; Schalch, Thomas; Chaplin, Amanda K

Molecular basis of pyruvate transport and inhibition of the human mitochondrial pyruvate carrier

丙酮酸转运的分子基础及人类线粒体丙酮酸载体的抑制

Sichrovsky, Maximilian; Lacabanne, Denis; Ruprecht, Jonathan J; Rana, Jessica J; Stanik, Klaudia; Dionysopoulou, Mariangela; Sowton, Alice P; King, Martin S; Jones, Scott A; Cooper, Lee; Hardwick, Steven W; Paris, Giulia; Chirgadze, Dimitri Y; Ding, Shujing; Fearnley, Ian M; Palmer, Shane M; Pardon, Els; Steyaert, Jan; Leone, Vanessa; Forrest, Lucy R; Tavoulari, Sotiria; Kunji, Edmund R S

High-Throughput Identification and Characterization of LptDE-Binding Bicycle Peptides Using Phage Display and Cryo-EM

利用噬菌体展示和冷冻电镜技术对LptDE结合双环肽进行高通量鉴定和表征

Allyjaun, Shenaz; Dunbar, Emily; Hardwick, Steven W; Newell, Sarah; Holding, Finn; Rowland, Catherine E; St Denis, Megan A; Pellegrino, Simone; Arruda Bezerra, Gustavo; Bournakas, Nikolaos; Chirgadze, Dimitri Y; Cooper, Lee; Paris, Giulia; Lewis, Nick; Brown, Peter; Skynner, Michael J; Dawson, Michael J; Beswick, Paul; Hubbard, Julia; van den Berg, Bert; Newman, Hector

Mechanism of NACHO-mediated assembly of pentameric ligand-gated ion channels

NACHO 介导五聚体配体门控离子通道组装的机制

Yogesh Hooda, Andrija Sente, Ryan M Judy, Luka Smalinskaitė, Sew-Yeu Peak-Chew, Katerina Naydenova, Tomas Malinauskas, Steven W Hardwick, Dimitri Y Chirgadze, A Radu Aricescu, Ramanujan S Hegde

Structural and functional basis of inositol hexaphosphate stimulation of NHEJ through stabilization of Ku-XLF interaction

肌醇六磷酸通过稳定 Ku-XLF 相互作用刺激 NHEJ 的结构和功能基础

Antonia Kefala Stavridi, Amandine Gontier, Vincent Morin, Philippe Frit, Virginie Ropars, Nadia Barboule, Carine Racca, Sagun Jonchhe, Michael J Morten, Jessica Andreani, Alexey Rak, Pierre Legrand, Alexa Bourand-Plantefol, Steven W Hardwick, Dimitri Y Chirgadze, Paul Davey, Taiana Maia De Oliveira,

The molecular basis of drug selectivity for α5 subunit-containing GABAA receptors

含α5亚基的GABAA受体药物选择性的分子基础

Vikram Babu Kasaragod, Tomas Malinauskas, Ayla A Wahid, Judith Lengyel, Frederic Knoflach, Steven W Hardwick, Charlotte F Jones, Wan-Na Chen, Xavier Lucas, Kamel El Omari, Dimitri Y Chirgadze, A Radu Aricescu, Giuseppe Cecere, Maria-Clemencia Hernandez, Paul S Miller

Structure of a bacterial ribonucleoprotein complex central to the control of cell envelope biogenesis

细菌核糖核蛋白复合物的结构对控制细胞膜生物合成至关重要

Md Saiful Islam, Steven W Hardwick, Laura Quell, Svetlana Durica-Mitic, Dimitri Y Chirgadze, Boris Görke, Ben F Luisi

Differential assembly diversifies GABAA receptor structures and signalling

差异组装使 GABAA 受体结构和信号传导多样化

Andrija Sente, Rooma Desai, Katerina Naydenova, Tomas Malinauskas, Youssef Jounaidi, Jonas Miehling, Xiaojuan Zhou, Simonas Masiulis, Steven W Hardwick, Dimitri Y Chirgadze, Keith W Miller, A Radu Aricescu

Mechanisms of inhibition and activation of extrasynaptic αβ GABAA receptors

突触外 αβ GABAA 受体的抑制和激活机制

Vikram Babu Kasaragod, Martin Mortensen, Steven W Hardwick, Ayla A Wahid, Valentina Dorovykh, Dimitri Y Chirgadze, Trevor G Smart, Paul S Miller