日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Direct GPCR-EGFR interaction enables synergistic membrane-to-nucleus information transfer

GPCR-EGFR直接相互作用可实现膜至细胞核的协同信息传递

Michael Gekle, Robert Eckenstaler, Heike Braun, Abdurrahman Olgac, Dina Robaa, Sigrid Mildenberger, Virginie Dubourg, Barbara Schreier, Wolfgang Sippl, Ralf Benndorf

Fatty acid binding to the human transport proteins FABP3, FABP4, and FABP5 from a Ligand's perspective

从配体角度看脂肪酸与人类运输蛋白 FABP3、FABP4 和 FABP5 的结合

Sebastian Michler, Florian Arndt Schöffmann, Dina Robaa, Jonas Volmer, Dariush Hinderberger

Identification of histone deacetylase 10 (HDAC10) inhibitors that modulate autophagy in transformed cells

鉴定调节转化细胞自噬的组蛋白去乙酰化酶 10 (HDAC10) 抑制剂

Patrik Zeyen, Yanira Zeyn, Daniel Herp, Fereshteh Mahmoudi, Talha Z Yesiloglu, Frank Erdmann, Matthias Schmidt, Dina Robaa, Christophe Romier, Johannes Ridinger, Corey J Herbst-Gervasoni, David W Christianson, Ina Oehme, Manfred Jung, Oliver H Krämer, Wolfgang Sippl

First Fluorescent Acetylspermidine Deacetylation Assay for HDAC10 Identifies Selective Inhibitors with Cellular Target Engagement

首次通过荧光乙酰亚精胺脱乙酰化试验鉴定出与细胞靶标结合的选择性抑制剂

Daniel Herp, Johannes Ridinger, Dina Robaa, Stephen A Shinsky, Karin Schmidtkunz, Talha Z Yesiloglu, Theresa Bayer, Raphael R Steimbach, Corey J Herbst-Gervasoni, Annika Merz, Christophe Romier, Peter Sehr, Nikolas Gunkel, Aubry K Miller, David W Christianson, Ina Oehme, Wolfgang Sippl, Manfred Jung

Design, Synthesis and Biological Characterization of Histone Deacetylase 8 (HDAC8) Proteolysis Targeting Chimeras (PROTACs) with Anti-Neuroblastoma Activity

具有抗神经母细胞瘤活性的组蛋白去乙酰化酶 8 (HDAC8) 蛋白水解靶向嵌合体 (PROTAC) 的设计、合成和生物学表征

Salma Darwish, Ehab Ghazy, Tino Heimburg, Daniel Herp, Patrik Zeyen, Rabia Salem-Altintas, Johannes Ridinger, Dina Robaa, Karin Schmidtkunz, Frank Erdmann, Matthias Schmidt, Christophe Romier, Manfred Jung, Ina Oehme, Wolfgang Sippl

Synthesis, Molecular Docking and Biological Characterization of Pyrazine Linked 2-Aminobenzamides as New Class I Selective Histone Deacetylase (HDAC) Inhibitors with Anti-Leukemic Activity

具有抗白血病活性的新型 I 类选择性组蛋白去乙酰化酶 (HDAC) 抑制剂吡嗪连接的 2-氨基苯甲酰胺的合成、分子对接和生物学表征

Hany S Ibrahim, Mohamed Abdelsalam, Yanira Zeyn, Matthes Zessin, Al-Hassan M Mustafa, Marten A Fischer, Patrik Zeyen, Ping Sun, Emre F Bülbül, Anita Vecchio, Frank Erdmann, Matthias Schmidt, Dina Robaa, Cyril Barinka, Christophe Romier, Mike Schutkowski, Oliver H Krämer, Wolfgang Sippl

Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma mansoni

药理学抑制赖氨酸特异性脱甲基酶 1 (LSD1) 会诱导整体转录失调和超微结构改变,从而损害曼氏血吸虫的生存能力

Vitor Coutinho Carneiro, Isabel Caetano de Abreu da Silva, Murilo Sena Amaral, Adriana S A Pereira, Gilbert Oliveira Silveira, David da Silva Pires, Sergio Verjovski-Almeida, Frank J Dekker, Dante Rotili, Antonello Mai, Eduardo José Lopes-Torres, Dina Robaa, Wolfgang Sippl, Raymond J Pierce, M Teres

Synthesis and Biological Investigation of Phenothiazine-Based Benzhydroxamic Acids as Selective Histone Deacetylase 6 Inhibitors

吩噻嗪类苯甲羟肟酸作为选择性组蛋白去乙酰化酶 6 抑制剂的合成及生物学研究

Katharina Vögerl, Nghia Ong, Johanna Senger, Daniel Herp, Karin Schmidtkunz, Martin Marek, Martin Müller, Karin Bartel, Tajith B Shaik, Nicholas J Porter, Dina Robaa, David W Christianson, Christophe Romier, Wolfgang Sippl, Manfred Jung, Franz Bracher

Chemically Induced Degradation of Sirtuin 2 (Sirt2) by a Proteolysis Targeting Chimera (PROTAC) Based on Sirtuin Rearranging Ligands (SirReals)

基于 Sirtuin 重排配体 (SirReals) 的蛋白水解靶向嵌合体 (PROTAC) 化学诱导 Sirtuin 2 (Sirt2) 降解

Matthias Schiedel, Daniel Herp, Sören Hammelmann, Sören Swyter, Attila Lehotzky, Dina Robaa, Judit Oláh, Judit Ovádi, Wolfgang Sippl, Manfred Jung

Selective agonist of TRPML2 reveals direct role in chemokine release from innate immune cells

TRPML2选择性激动剂揭示其在固有免疫细胞趋化因子释放中的直接作用

Eva Plesch # ,Cheng-Chang Chen # ,Elisabeth Butz # ,Anna Scotto Rosato ,Einar K Krogsaeter ,Hua Yinan ,Karin Bartel ,Marco Keller ,Dina Robaa ,Daniel Teupser ,Lesca M Holdt ,Angelika M Vollmar ,Wolfgang Sippl ,Rosa Puertollano ,Diego Medina ,Martin Biel ,Christian Wahl-Schott ,Franz Bracher ,Christian Grimm