日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The electrophilic metabolite of kynurenine, kynurenine-CKA, requires C151 in Keap1 to derepress Nrf2

犬尿氨酸的亲电代谢产物犬尿氨酸-CKA需要Keap1中的C151才能解除Nrf2的抑制。

Feng, Jialin; Carreño, Mara; Jung, Hannah; Dayalan Naidu, Sharadha; Arroyo-Diaz, Nicole; Ang, Abel D; Kulkarni, Bhargavi; Kisielewski, Dorothy; Suzuki, Takafumi; Yamamoto, Masayuki; Hayes, John D; Honda, Tadashi; Wilson, Landon; Leon-Ruiz, Beatriz; Eggler, Aimee L; Vitturi, Dario A; Dinkova-Kostova, Albena T

Keap1-Kelch-targeting protein-protein interaction inhibitors, but not reversibly-binding electrophiles, increase the thermostability of Keap1 in the cellular environment

靶向Keap1-Kelch的蛋白质-蛋白质相互作用抑制剂,而非可逆结合的亲电试剂,能够提高Keap1在细胞环境中的热稳定性。

Dayalan Naidu, Sharadha; Dikovskaya, Dina; Walker, Jasmine M; Yee, Charlotte Lim Jia; Cafferkey, Annamarie J; Tatsuno, Manaka; Feng, Jialin; Moore, Terry W; Johnson, Tatum; Honda, Tadashi; Wells, Geoff; Suzuki, Takafumi; Yamamoto, Masayuki; Dinkova-Kostova, Albena T

The tasiR-ARF pathway in plants: origin, functions, and interplay of miR-390, tasiRNAs and ARF3

植物中的 tasiR-ARF 通路:miR-390、tasiRNA 和 ARF3 的起源、功能和相互作用

López-Ruiz, B A; Juárez González, V T; Jiménez-Ortega, R F; Reyes, J L; Dinkova, T D

M102 activates both NRF2 and HSF1 transcription factor pathways and is neuroprotective in cell and animal models of amyotrophic lateral sclerosis

M102 可激活 NRF2 和 HSF1 转录因子通路,并在肌萎缩侧索硬化症的细胞和动物模型中发挥神经保护作用。

Keerie, Amy F; Martins, Raquel Rua; Allen, Chloe F; Bowden, Katie; Al Mashhadi, Sufana; Marlow, Thomas; Myszczynska, Monika; Thakur, Nikitha; Beal, Selina N; Shaw, Allan; Suresh, Shivani; McKinnon, Scott N; Cooper-Knock, Johnathan; West, Ryan J H; Bonsall, Sam; Daniel, Alex; Wells, Tyler; Kumar, Vedanth; Ellis, Brittany C S; Higgins, Maureen; Dinkova-Kostova, Albena T; Shelkovnikova, Tatyana A; Kalfus, Ira N; Shan, Ning; Shaw, Pamela J; Ferraiuolo, Laura; Mead, Richard J

Model organisms for investigating the functional involvement of NRF2 in non-communicable diseases

用于研究 NRF2 在非传染性疾病中功能作用的模式生物

Rojo, Ana I; Buttari, Brigitta; Cadenas, Susana; Carlos, Ana Rita; Cuadrado, Antonio; Falcão, Ana Sofia; López, Manuela G; Georgiev, Milen I; Grochot-Przeczek, Anna; Gumeni, Sentiljana; Jimenez-Villegas, José; Horbanczuk, Jarosław Olav; Konu, Ozlen; Lastres-Becker, Isabel; Levonen, Anna-Liisa; Maksimova, Viktorija; Michaeloudes, Charalambos; Mihaylova, Liliya V; Mickael, Michel Edwar; Milisav, Irina; Miova, Biljana; Rada, Patricia; Santos, Marlene; Seabra, Miguel C; Strac, Dubravka Svob; Tenreiro, Sandra; Trougakos, Ioannis P; Dinkova-Kostova, Albena T

Corrigendum to "Model organisms for investigating the functional involvement of NRF2 in non-communicable diseases" [Redox Biol. 79 (2025) 103464]

对“用于研究 NRF2 在非传染性疾病中的功能作用的模型生物”的更正 [Redox Biol. 79 (2025) 103464]

Rojo, Ana I; Buttari, Brigitta; Cadenas, Susana; Carlos, Ana Rita; Cuadrado, Antonio; Falcão, Ana Sofia; López, Manuela G; Georgiev, Milen I; Grochot-Przeczek, Anna; Gumeni, Sentiljana; Jiménez-Villegas, José; Horbanczuk, Jarosław Olav; Konu, Ozlen; Lastres-Becker, Isabel; Levonen, Anna-Liisa; Maksimova, Viktorija; Michaeloudes, Charalambos; Mihaylova, Liliya V; Mickael, Michel Edwar; Milisav, Irina; Miova, Biljana; Rada, Patricia; Santos, Marlene; Seabra, Miguel C; Strac, Dubravka Svob; Tenreiro, Sandra; Trougakos, Ioannis P; Dinkova-Kostova, Albena T

Health position paper and redox perspectives - Bench to bedside transition for pharmacological regulation of NRF2 in noncommunicable diseases

健康立场文件和氧化还原视角——非传染性疾病中NRF2药物调控的从实验室到临床转化

Cuadrado, Antonio; Cazalla, Eduardo; Bach, Anders; Bathish, Boushra; Naidu, Sharadha Dayalan; DeNicola, Gina M; Dinkova-Kostova, Albena T; Fernández-Ginés, Raquel; Grochot-Przeczek, Anna; Hayes, John D; Kensler, Thomas W; León, Rafael; Liby, Karen T; López, Manuela G; Manda, Gina; Shivakumar, Akshatha Kalavathi; Hakomäki, Henriikka; Moerland, Jessica A; Motohashi, Hozumi; Rojo, Ana I; Sykiotis, Gerasimos P; Taguchi, Keiko; Valverde, Ángela M; Yamamoto, Masayuki; Levonen, Anna-Liisa

Tetrazole-containing naphthalene bis-sulfonamide Keap1-Nrf2 interaction inhibitors with unexpected binding modes.

具有意想不到的结合模式的含四唑萘双磺酰胺 Keap1-Nrf2 相互作用抑制剂。

Georgakopoulos Nikolaos D, Talapatra Sandeep K, Dayalan Naidu Sharadha, Dikovskaya Dina, Higgins Maureen, Gatliff Jemma, Nikoloudaki Roxani, Schaap Marjolein, Walker Jasmine M, Wardby Christopher, Dinkova-Kostova Albena T, Harris Sarah, Kozielski Frank, Wells Geoff

Activation of the Nrf2 Pathway by Sulforaphane Improves Hypoglycaemia-Induced Cognitive Impairment in a Rodent Model of Type 1 Diabetes

萝卜硫素激活Nrf2通路可改善1型糖尿病啮齿动物模型中低血糖引起的认知障碍

Merchant, Heather J; Forteath, Calum; Gallagher, Jennifer R; Dinkova-Kostova, Albena T; Ashford, Michael L J; McCrimmon, Rory J; McNeilly, Alison D

Genetic Deletion of RHAMM Alleviates Hepatic Oxidative Stress, Reversing Thyroid Stimulating Hormone Elevation in Male Obese Mice

RHAMM基因缺失可减轻雄性肥胖小鼠的肝脏氧化应激,逆转促甲状腺激素水平升高

Wang, Tianzhen; Sun, Helin; Banah, Ayman K; Weng, Xiong; Dayalan Naidu, Sharadha; Kisielewski, Dot; Ang, Abel; Hayes, John D; Dinkova-Kostova, Albena T; Kang, Li