日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Chemical Modification of Pactamycin Leads to New Compounds with Retained Antimicrobial Activity and Reduced Toxicity

帕克他霉素的化学修饰可得到保留抗菌活性且毒性降低的新化合物

Tsirogianni, Artemis; Ntinou, Nikolina; Karampatsou, Konstantina; Dinos, George; Kournoutou, Georgia G; Athanassopoulos, Constantinos M

Chloramphenicol Derivatization in Its Primary Hydroxyl Group with Basic Amino Acids Leads to New Pharmacophores with High Antimicrobial Activity.

氯霉素伯羟基与碱性氨基酸衍生化,可得到具有高抗菌活性的新型药效团

Tsirogianni Artemis, Kournoutou Georgia G, Mpogiatzoglou Maria, Dinos George, Athanassopoulos Constantinos M

Azithromycin through the Lens of the COVID-19 Treatment

从新冠肺炎治疗的角度看阿奇霉素

Kournoutou, Georgia G; Dinos, George

New Chloramphenicol Derivatives with a Modified Dichloroacetyl Tail as Potential Antimicrobial Agents.

具有修饰的二氯乙酰尾的新型氯霉素衍生物作为潜在的抗菌剂

Tsirogianni Artemis, Kournoutou Georgia G, Bougas Anthony, Poulou-Sidiropoulou Eleni, Dinos George, Athanassopoulos Constantinos M

High-resolution crystal structures of ribosome-bound chloramphenicol and erythromycin provide the ultimate basis for their competition

核糖体结合的氯霉素和红霉素的高分辨率晶体结构为它们之间的竞争提供了最终依据。

Svetlov, Maxim S; Plessa, Elena; Chen, Chih-Wei; Bougas, Anthony; Krokidis, Marios G; Dinos, George P; Polikanov, Yury S

New Chloramphenicol Derivatives from the Viewpoint of Anticancer and Antimicrobial Activity

从抗癌和抗菌活性角度看新型氯霉素衍生物

Giannopoulou, Panagiota C; Missiri, Dionissia A; Kournoutou, Georgia G; Sazakli, Eleni; Papadopoulos, Georgios E; Papaioannou, Dionissios; Dinos, George P; Athanassopoulos, Constantinos M; Kalpaxis, Dimitrios L

Chloramphenicol Derivatives as Antibacterial and Anticancer Agents: Historic Problems and Current Solutions

氯霉素衍生物作为抗菌和抗癌药物:历史问题与当前解决方案

Dinos, George P; Athanassopoulos, Constantinos M; Missiri, Dionissia A; Giannopoulou, Panagiota C; Vlachogiannis, Ioannis A; Papadopoulos, Georgios E; Papaioannou, Dionissios; Kalpaxis, Dimitrios L

Linezolid-dependent function and structure adaptation of ribosomes in a Staphylococcus epidermidis strain exhibiting linezolid dependence.

对利奈唑胺有依赖性的表皮葡萄球菌菌株中核糖体的利奈唑胺依赖性功能和结构适应性

Kokkori Sofia, Apostolidi Maria, Tsakris Athanassios, Pournaras Spyros, Stathopoulos Constantinos, Dinos George

Distinct mode of interaction of a novel ketolide antibiotic that displays enhanced antimicrobial activity

一种新型酮内酯类抗生素具有独特的相互作用模式,并表现出增强的抗菌活性。

Kouvela, Ekaterini C; Kalpaxis, Dimitrios L; Wilson, Daniel N; Dinos, George P

Effect of polyamines on the inhibition of peptidyltransferase by antibiotics: revisiting the mechanism of chloramphenicol action.

多胺对抗生素抑制肽基转移酶的影响:重新审视氯霉素的作用机制

Xaplanteri Maria A, Andreou Athanasios, Dinos George P, Kalpaxis Dimitrios L