日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Chromones as Nonclassical Inhibitors of Carbonic Anhydrase IX and XII Isoforms: Probing Chromone-Based Derivatives

色酮类化合物作为碳酸酐酶IX和XII同工酶的非经典抑制剂:探索基于色酮的衍生物

Sequeira, Lisa; Distinto, Simona; Fernandes, Carlos; Sanna, Erica; Meleddu, Rita; Gaspari, Marco; Cottiglia, Filippo; Onali, Alessia; Angeli, Andrea; Borges, Fernanda; Uriarte, Eugenio; Alcaro, Stefano; Supuran, Claudiu T; Maccioni, Elias

Synthesis and Evaluation of Thiazolidinone-Isatin Hybrids for Selective Inhibition of Cancer-Related Carbonic Anhydrases

噻唑烷酮-靛红杂合物的合成与评价及其对癌症相关碳酸酐酶的选择性抑制作用

Onali, Alessia; Sanna, Erica; Lupia, Antonio; Secci, Daniela; Atzeni, Giulia; Demuru, Laura; Angeli, Andrea; Cottiglia, Filippo; Meleddu, Rita; Emmolo, Roberta; Corona, Angela; Maccioni, Elias; Supuran, Claudiu T; Distinto, Simona

Privileged Scaffold Hybridization in the Design of Carbonic Anhydrase Inhibitors

碳酸酐酶抑制剂设计中的特权支架杂交

Daniela Secci, Erica Sanna, Simona Distinto, Alessia Onali, Antonio Lupia, Laura Demuru, Giulia Atzeni, Rita Meleddu, Filippo Cottiglia, Andrea Angeli, Claudiu T Supuran, Elias Maccioni

Identification of new benzofuran derivatives as STING agonists with broad-spectrum antiviral activity

鉴定具有广谱抗病毒活性的新型苯并呋喃衍生物作为 STING 激动剂

A Paulis, A Onali, P O Vidalain, V Lotteau, C Jaquemin, A Corona, S Distinto, G L Delogu, E Tramontano

5-Nitro-3-(2-(4-phenylthiazol-2-yl)hydrazineylidene)indolin-2-one derivatives inhibit HIV-1 replication by a multitarget mechanism of action

5-硝基-3-(2-(4-苯基噻唑-2-基)肼基亚甲基)吲哚啉-2-酮衍生物通过多靶点作用机制抑制HIV-1复制

Corona, Angela; Meleddu, Rita; Delelis, Olivier; Subra, Frederic; Cottiglia, Filippo; Esposito, Francesca; Distinto, Simona; Maccioni, Elias; Tramontano, Enzo

Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase-associated RNase H function

来自黄毛香科植物(Teucrium flavum subsp. glaucum)的黄酮类化合物和新克罗丹二萜酸水解衍生物作为HIV-1逆转录酶相关RNase H功能的抑制剂

Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo

2-(2-Methyl-2-nitrovinyl)furan but Not Furvina Interfere with Staphylococcus aureus Agr Quorum-Sensing System and Potentiate the Action of Fusidic Acid against Biofilms

2-(2-甲基-2-硝基乙烯基)呋喃而非呋喃酮干扰金黄色葡萄球菌Agr群体感应系统并增强夫西地酸对生物膜的作用

Oliveira, Diana; Borges, Anabela; Ruiz, Reinaldo Molina; Negrín, Zenaida Rodríguez; Distinto, Simona; Borges, Fernanda; Simões, Manuel

Quercetin Blocks Ebola Virus Infection by Counteracting the VP24 Interferon-Inhibitory Function

槲皮素通过抵消 VP24 干扰素抑制功能来阻止埃博拉病毒感染

Elisa Fanunza, Mathieu Iampietro, Simona Distinto, Angela Corona, Marina Quartu, Elias Maccioni, Branka Horvat, Enzo Tramontano

Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 reverse transcriptase-associated RNase H and RDDP functions

设计、合成并评价新型杂芳基硫代甲酰胺衍生物作为HIV-1逆转录酶相关RNase H和RDDP功能的双重抑制剂的抗病毒活性

Corona, Angela; Onnis, Valentina; Deplano, Alessandro; Bianco, Giulia; Demurtas, Monica; Distinto, Simona; Cheng, Yung-Chi; Alcaro, Stefano; Esposito, Francesca; Tramontano, Enzo

Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors

环庚噻吩-3-甲酰胺衍生物作为变构HIV-1核糖核酸酶H抑制剂的研究

Corona, Angela; Desantis, Jenny; Massari, Serena; Distinto, Simona; Masaoka, Takashi; Sabatini, Stefano; Esposito, Francesca; Manfroni, Giuseppe; Maccioni, Elias; Cecchetti, Violetta; Pannecouque, Christophe; Le Grice, Stuart F J; Tramontano, Enzo; Tabarrini, Oriana