Discovery of Potent and Selective 7-Azaindole Isoindolinone-Based PI3Kγ Inhibitors
发现高效选择性的7-氮杂吲哚异吲哚啉酮类PI3Kγ抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.0c00387
Miles, Dillon H; Yan, Xuelei; Thomas-Tran, Rhiannon; Fournier, Jeremy; Sharif, Ehesan U; Drew, Samuel L; Mata, Guillaume; Lawson, Kenneth V; Ginn, Elaine; Wong, Kent; Soni, Divyank; Dhanota, Puja; Shaqfeh, Stefan G; Meleza, Cesar; Chen, Ada; Pham, Amber T; Park, Timothy; Swinarski, Debbie; Banuelos, Jesus; Schindler, Ulrike; Walters, Matthew J; Walker, Nigel P; Zhao, Xiaoning; Young, Stephen W; Chen, Jie; Jin, Lixia; Leleti, Manmohan Reddy; Powers, Jay P; Jeffrey, Jenna L