日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a peptide proteolysis-targeting chimera (PROTAC) drug of p300 for prostate cancer therapy

发现一种靶向p300肽蛋白水解的嵌合体(PROTAC)药物用于前列腺癌治疗

Dize Zhang,Bohan Ma,Donghua Liu,Wei Wu,Tianyang Zhou,Yibo Gao,Cunli Yang,Yanlin Jian,Yizeng Fan,Yuchen Qian,Jian Ma,Yang Gao,Yule Chen,Shan Xu,Lei Li

Development of a Double-Stapled Peptide Stabilizing Both α-Helix and β-Sheet Structures for Degrading Transcription Factor AR-V7

开发稳定 α-螺旋和 β-片层结构的双钉肽,用于降解转录因子 AR-V7

Bohan Ma, Donghua Liu, Mengjun Zheng, Zhe Wang, Dize Zhang, Yanlin Jian, Jian Ma, Yizeng Fan, Yule Chen, Yang Gao, Jing Liu, Xiang Li, Lei Li

De Novo Design of an Androgen Receptor DNA Binding Domain-Targeted peptide PROTAC for Prostate Cancer Therapy

针对雄激素受体 DNA 结合域的肽 PROTAC 的从头设计,用于前列腺癌治疗

Bohan Ma, Yizeng Fan, Dize Zhang, Yi Wei, Yanlin Jian, Donghua Liu, Zixi Wang, Yang Gao, Jian Ma, Yule Chen, Shan Xu, Lei Li