日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

l‑Boronophenylalanine (l-BPA) Dipeptide Prodrugs Enhance Boron Delivery to Tumors, Facilitate Tumor Eradication and Induce Tumor Vaccine Effect in Mice Following Neutron Irradiation.

l-硼苯丙氨酸(l-BPA)二肽前药可增强硼向肿瘤的输送,促进肿瘤根除,并在中子照射后诱导小鼠肿瘤疫苗效应。

Torgov Michael, Raitano Arthur, Quintana Jason Cole, Martin Tioga, Kulenovic Leila, Dlamini Samkeliso, Zhang Chunying, Malinao Maria-Christina, Ikeura Maki, Capo Linnette, Morrison Karen, Matsumoto Kotaro, Komatsu Aoi, Higashi Yuya, Takushi Takata, Sakurai Yoshinori, Dorn Robert, Suzuki Minoru, Tamanoi Fuyuhiko, Morrison Kendall

Regulation of ferroptosis by transcription factor E2F1.

转录因子E2F1调控铁死亡

Kuganesan Nishanth, Dlamini Samkeliso, Hasan Safiyyah, Viranga Tillekeratne L M, Taylor William R

CETZOLE Analogs as Potent Ferroptosis Inducers and Their Target Identification Using Covalent/Affinity Probes.

CETZOLE 类似物作为强效铁死亡诱导剂及其利用共价/亲和探针进行靶标鉴定

Dlamini Samkeliso, Mohajeri Shahrzad, Kuganesan Nishanth, Sindi Shaimaa H, Karaj Endri, Rathnayake Dewmi S, McDaniel Jade, Taylor William R, Tillekeratne L M Viranga

Pharmacophore optimization of imidazole chalcones to modulate microtubule dynamics

利用咪唑查尔酮的药效团优化来调节微管动力学

Karaj, Endri; Dlamini, Samkeliso; Koranne, Radhika; Sindi, Shaimaa H; Perera, Lalith; Taylor, William R; Viranga Tillekeratne, L M

Synthesis and Development of a Novel First-in-Class Cofilin Inhibitor for Neuroinflammation in Hemorrhagic Brain Injury.

合成和开发一种新型首创的cofilin抑制剂用于治疗出血性脑损伤引起的神经炎症

Alaqel Saleh I, Dlamini Samkeliso, Almarghalani Daniyah A, Shettigar Arjun, Alhadidi Qasim, Kodithuwakku Sinali H, Stary Creed, Tillekeratne L M Viranga, Shah Zahoor A