日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of Prostate-Specific Membrane Antigen-Targeted Bimodal Conjugates of Cytotoxic Agents and Antiandrogens and Their Comparative Assessment with Monoconjugates

前列腺特异性膜抗原靶向细胞毒剂和抗雄激素双峰结合物的合成及其与单结合物的比较评估

Nikolai Y Zyk, Anastasiia S Garanina, Ekaterina A Plotnikova, Anton P Ber, Ekaterina A Nimenko, Natalia S Dashkova, Anastasiia A Uspenskaia, Radik R Shafikov, Dmitry A Skvortsov, Stanislav A Petrov, Andrey A Pankratov, Nikolai V Zyk, Alexander G Majouga, Elena K Beloglazkina, Aleksei E Machulkin

Copper coordination compounds with (5 Z,5 Z')-2,2'-(alkane-α,ω-diyldiselenyl)-bis-5-(2-pyridylmethylene)-3,5-dihydro-4 H-imidazol-4-ones. Comparison with sulfur analogue

铜与 (5 Z,5 Z')-2,2'-(烷-α,ω-二基二硒基)-双-5-(2-吡啶基亚甲基)-3,5-二氢-4 H-咪唑-4-酮的配位化合物。与硫类似物的比较

Alexander V Finko, Anatolii I Sokolov, Dmitry A Guk, Victor A Tafeenko, Anna A Moiseeva, Dmitry A Skvortsov, Andrei A Stomakhin, Andrei A Beloglazkin, Roman S Borisov, Vladimir I Pergushov, Mikhail Ya Melnikov, Nikolay V Zyk, Alexander G Majouga, Elena K Beloglazkina

Conjugates of Chloramphenicol Amine and Berberine as Antimicrobial Agents

氯霉素胺与小檗碱结合物的抗菌作用

Julia A Pavlova, Andrey G Tereshchenkov, Pavel A Nazarov, Dmitrii A Lukianov, Dmitry A Skvortsov, Vladimir I Polshakov, Byasilya F Vasilieva, Olga V Efremenkova, Mikhail Y Kaiumov, Alena Paleskava, Andrey L Konevega, Olga A Dontsova, Ilya A Osterman, Alexey A Bogdanov, Natalia V Sumbatyan

Dispirooxindoles Based on 2-Selenoxo-Imidazolidin-4-Ones: Synthesis, Cytotoxicity and ROS Generation Ability

基于 2-硒氧咪唑烷-4-酮的二吡咯吲哚:合成、细胞毒性和 ROS 生成能力

Vladimir K Novotortsev, Maxim E Kukushkin, Viktor A Tafeenko, Dmitry A Skvortsov, Marina A Kalinina, Roman V Timoshenko, Nelly S Chmelyuk, Liliya A Vasilyeva, Boris N Tarasevich, Petr V Gorelkin, Alexander S Erofeev, Alexander G Majouga, Nikolai V Zyk, Elena K Beloglazkina

Triphenilphosphonium Analogs of Chloramphenicol as Dual-Acting Antimicrobial and Antiproliferating Agents

氯霉素的三苯膦类似物作为双重抗菌和抗增殖剂

Julia A Pavlova, Zimfira Z Khairullina, Andrey G Tereshchenkov, Pavel A Nazarov, Dmitrii A Lukianov, Inna A Volynkina, Dmitry A Skvortsov, Gennady I Makarov, Etna Abad, Somay Y Murayama, Susumu Kajiwara, Alena Paleskava, Andrey L Konevega, Yuri N Antonenko, Alex Lyakhovich, Ilya A Osterman, Alexey A

Amicoumacin A induces cancer cell death by targeting the eukaryotic ribosome

Amicoumacin A 通过靶向真核核糖体诱导癌细胞死亡

Irina V Prokhorova, Kseniya A Akulich, Desislava S Makeeva, Ilya A Osterman, Dmitry A Skvortsov, Petr V Sergiev, Olga A Dontsova, Gulnara Yusupova, Marat M Yusupov, Sergey E Dmitriev