Selective inhibition of EZH2 and EZH1 enzymatic activity by a small molecule suppresses MLL-rearranged leukemia
小分子选择性抑制EZH2和EZH1酶活性可抑制MLL重排白血病。
期刊:Blood
影响因子:23.1
doi:10.1182/blood-2014-06-581082
Xu, Bowen; On, Doan M; Ma, Anqi; Parton, Trevor; Konze, Kyle D; Pattenden, Samantha G; Allison, David F; Cai, Ling; Rockowitz, Shira; Liu, Shichong; Liu, Ying; Li, Fengling; Vedadi, Masoud; Frye, Stephen V; Garcia, Benjamin A; Zheng, Deyou; Jin, Jian; Wang, Gang Greg