日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Disarming carbapenemase-producing Acinetobacter baumannii: high potency of the novel therapeutic combination of meropenem and the innovative diazabicyclooctane β-lactamase inhibitor pilabactam (formerly ANT3310)

解除产碳青霉烯酶鲍曼不动杆菌的毒力:美罗培南与创新型二氮杂双环辛烷β-内酰胺酶抑制剂匹拉巴坦(原名ANT3310)的新型治疗组合具有高效性

Rodríguez-Pallares, Salud; Outeda-García, Michelle; Lence, Emilio; Rodríguez-Coello, Arianna; González-Pinto, Lucía; Guijarro-Sánchez, Paula; Báez-Barroso, Gabriela Alejandra; Blanco-Martín, Tania; Vázquez-Ucha, Juan Carlos; Llanos, Agustina; Sannio, Filomena; Docquier, Jean-Denis; Morrisey, Ian; Hawser, Stephen; Zalacain, Magdalena; Lemonnier, Marc; González-Bello, Concepción; Bou, Germán; Beceiro, Alejandro; Arca-Suárez, Jorge

Oxyprenyl-chalcones as antibacterial hits: design of experiments-optimized synthesis, antibacterial evaluation, early drug-like profiling and biodegradability prediction

氧异戊烯基查尔酮类化合物作为抗菌先导化合物:实验设计优化合成、抗菌活性评价、早期类药性分析和生物降解性预测

Marotta, Ludovica; Giammarino, Francesca Maria Pia Rita; Senenou Tambou, Brondon Brandly; Tudino, Valeria; Butini, Stefania; Broccardo, Lorenza; Cancade, Sacha Michèle Idriss; Docquier, Jean-Denis; Perego, Federica; Basilico, Nicoletta; Raffellini, Lorenzo; Gul, Sheraz; Carullo, Gabriele; Gemma, Sandra; Campiani, Giuseppe

Sustainable Joullié-Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors.

可持续的 Joullié-Ugi 和连续流实施产生了新型的受卡托普利启发的广谱金属β-内酰胺酶抑制剂

Alfano Antonella Ilenia, Pelliccia Sveva, Barone Simona, Cutarella Luigi, Cancade Sacha Michèle Idriss, Baia Valerio, Cassese Emilia, Russomanno Pasquale, Messano Nicolò, Frank Denia, Weizel Lilia, Rotter Marco J, Brunst Steffen, Wichelhaus Thomas A, Proschak Ewgenij, Tedesco Daniele, Mori Mattia, Docquier Jean Denis, Summa Vincenzo, Brindisi Margherita

SAND: a comprehensive annotation of class D β-lactamases using structural alignment-based numbering

SAND:基于结构比对编号的D类β-内酰胺酶的综合注释

Attana, Fedaa; Kim, Soobin; Spencer, James; Iorga, Bogdan I; Docquier, Jean-Denis; Rossolini, Gian Maria; Perilli, Mariagrazia; Amicosante, Gianfranco; Vila, Alejandro J; Vakulenko, Sergei B; Mobashery, Shahriar; Bradford, Patricia; Bush, Karen; Partridge, Sally R; Hujer, Andrea M; Hujer, Kristine M; Bonomo, Robert A; Haider, Shozeb

Chaetomorpha linum Extract as a Source of Antimicrobial Compounds: A Circular Bioeconomy Approach

亚麻毛壳菌提取物作为抗菌化合物来源:一种循环生物经济方法

Barletta, Roberta; Trezza, Alfonso; Geminiani, Michela; Frusciante, Luisa; Olmastroni, Tommaso; Sannio, Filomena; Docquier, Jean-Denis; Santucci, Annalisa

4-Trifluoromethyl bithiazoles as broad-spectrum antimicrobial agents for virus-related bacterial infections or co-infections

4-三氟甲基联噻唑类化合物作为广谱抗菌剂用于治疗病毒相关细菌感染或合并感染

Barbieri, Francesca; Carlen, Vincent; Martina, Maria Grazia; Sannio, Filomena; Cancade, Sacha; Perini, Cecilia; Restori, Margherita; Crespan, Emmanuele; Maga, Giovanni; Docquier, Jean-Denis; Cagno, Valeria; Radi, Marco

Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships

苯磺酰胺衍生物作为霍乱弧菌碳酸酐酶抑制剂:计算辅助揭示结构刚性与活性关系

Fantacuzzi, Marialuigia; D'Agostino, Ilaria; Carradori, Simone; Liguori, Francesco; Carta, Fabrizio; Agamennone, Mariangela; Angeli, Andrea; Sannio, Filomena; Docquier, Jean-Denis; Capasso, Clemente; Supuran, Claudiu T

Peptaibol Analogs Show Potent Antibacterial Activity against Multidrug Resistant Opportunistic Pathogens

肽类化合物类似物对多重耐药机会性病原体表现出强效抗菌活性

Dalla Torre, Chiara; Sannio, Filomena; Battistella, Mattia; Docquier, Jean-Denis; De Zotti, Marta

Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors

发现和优化新型大环脒基脲系列化合物,该系列化合物可作为酸性哺乳动物几丁质酶抑制剂

Balestri, Lorenzo Jacopo Ilic; Trivisani, Claudia Immacolata; Orofino, Francesco; Fiorucci, Diego; Truglio, Giuseppina Ivana; D'Agostino, Ilaria; Poggialini, Federica; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena

Discovering NDM-1 inhibitors using molecular substructure embeddings representations

利用分子亚结构嵌入表示法发现NDM-1抑制剂

Papastergiou, Thomas; Azé, Jérôme; Bringay, Sandra; Louet, Maxime; Poncelet, Pascal; Rosales-Hurtado, Miyanou; Vo-Hoang, Yen; Licznar-Fajardo, Patricia; Docquier, Jean-Denis; Gavara, Laurent