日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Evaluating Acridones as Novel Therapeutics for Human Babesiosis

评估吖啶酮类化合物作为治疗人类巴贝虫病的新型疗法

Vydyam, Pratap; Zhang, Elizabeth; Pal, Anasuya C; Dodean, Rozalia A; Kancharla, Papireddy; Kelly, Jane X; Ben Mamoun, Choukri

Optimization of Prodiginines as Single-Dose Curative Antimalarials

优化灵菌红素类药物作为单剂量治愈性抗疟药

Kumar, Amrendra; Li, Yuexin; Zhang, Xiaowei; Gaddam, Mahesh; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Chetree, Ravi; Blount, Cameron; DeLuca, Jesse; Vuong, Chau; Kudyba, Karl; Roncal, Norma; Ashraf, Kutub; Lee, Patricia J; Pannone, Kristina; Leed, Susan; Dinh, Hieu T; Mdaki, Kennedy; Navarrete, Kimberly; Charlton, Jordan; Binauhan, Angely J; Qahash, Tarrick; Kibe, Kevin Mugambi; Shoue, Douglas A; Checkley, Lisa; Ferdig, Michael T; Chim-Ong, Anongruk; Cui, Liwang; Orena, Stephen; Byaruhanga, Oswald; Assimwe, Jackson; Tibagambirwa, Innocent; Chithanna, Sivanna; Dodean, Rozalia A; Legac, Jennifer; Kreutzfeld, Oriana; Rosenthal, Philip J; Cooper, Roland A; Reynolds, Kevin A; Roth, Alison; Kelly, Jane X; Kancharla, Papireddy

Acridone Prodrugs with Enhanced Dual-Stage Antimalarial Efficacy

具有增强双阶段抗疟功效的吖啶酮前药

Dodean, Rozalia A; Li, Yuexin; Zhang, Xiaowei; Kumar, Amrendra; Pou, Sovitj; W Winter, Rolf; Liebman, Katherine M; Zakharov, Lev N; Caridha, Diana; Madejczyk, Michael S; Vuong, Chau; DeLuca, Jesse; Chin, Geoffrey; Kudyba, Karl; McEnearney, Sharon; Jin, Xiannu; Dennis, William E; Chetree, Ravi; Blount, Cameron; Pannone, Kristina; Dinh, Hieu T; Mdaki, Kennedy; Leed, Susan; Lee, Patricia J; Roth, Alison; Kancharla, Papireddy; Kelly, Jane X

Identifying antimalarials that disrupt malaria parasite transmission when fed to the mosquito

鉴定出喂给蚊子后能阻断疟原虫传播的抗疟药。

Farrell, Sarah N; Cozijnsen, Anton; Mollard, Vanessa; Kancharla, Papireddy; Dodean, Rozalia A; Kelly, Jane X; McFadden, Geoffrey I; Goodman, Christopher D

Potent Acridone Antimalarial against All Three Life Stages of Plasmodium

强效抗疟药吖啶酮,可对抗疟原虫所有三个生命阶段

Kancharla, Papireddy; Dodean, Rozalia A; Li, Yuexin; Zhang, Xiaowei; Kelly, Sean; Charlton, Jordan; Binauhan, Angley; Garcia, Laurize; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Kudyba, Karl; McEnearney, Sharon; Lee, Partricia J; Blount, Cameron; DeLuca, Jesse; Vuong, Chua; Pannone, Kristina; Dinh, Hieu T; Mdaki, Kennedy; Leed, Susan; Martin, Monica L; Pybus, Brandon S; Chimong, Anongruk; Cui, Liwang; Vega-Rodriguez, Joel; Okitwi, Martin; Kreutzfeld, Oriana; Docan, Christina; Green, Carol; Liu, Ying; Agulay, Aaron; Mirsalis, Jon; Farrell, Sarah N; McFadden, Geoffrey I; Goodman, Christopher D; Probst, Alexandra S; Nilsen, Aaron; Catteruccia, Flaminia; Rosenthal, Philip J; Riscoe, Michael; Cooper, Roland; Roth, Alison; Kelly, Jane

Discovery and Optimization of Tambjamines as a Novel Class of Antileishmanial Agents

发现和优化 Tambjamines 作为一类新型抗利什曼原虫药物

Papireddy Kancharla, Diana Ortiz, Corinne M Fargo, Xiaowei Zhang, Yuexin Li, Marco Sanchez, Amrendra Kumar, Monish Yeluguri, Rozalia A Dodean, Diana Caridha, Michael S Madejczyk, Monica Martin, Xiannu Jin, Cameron Blount, Ravi Chetree, Kristina Pannone, Hieu T Dinh, Jesse DeLuca, Martin Evans, Rober

Long-acting intramuscular injections of ELQ-331, an antimalarial agent

长效肌注抗疟药ELQ-331

Karunakaran, Dipu; Mutyam, Shravan K; Fu, Melody; Chen, Jiaming; Pham, Kim Hue Nicky; Pou, Sovitj; Winter, Rolf W; Nilsen, Aaron; Dodean, Rozalia A; Smilkstein, Martin J; Riscoe, Michael K; Shankar, Gita

DDDR-05. SPATIALLY RESOLVED DRUG SENSITIVITY PROFILING IN GLIOBLASTOMA

DDDR-05. 胶质母细胞瘤的空间分辨药物敏感性分析

Kumar, Amrendra; Li, Yuexin; Dodean, Rozalia A; Roth, Alison; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Lee, Patricia J; Pybus, Brandon S; Martin, Monica; Pannone, Kristina; Dinh, Hieu T; Blount, Cameron; Chetree, Ravi; DeLuca, Jesse; Evans, Martin; Nadeau, Robert; Vuong, Chau; Leed, Susan; Black, Chad; Sousa, Jason; Nolan, Christina; Ceja, Frida G; Rasmussen, Stephanie A; Tumwebaze, Patrick K; Rosenthal, Philip J; Cooper, Roland A; Rottmann, Matthias; Orjuela-Sanchez, Pamela; Meister, Stephan; Winzeler, Elizabeth A; Delves, Michael J; Matthews, Holly; Baum, Jake; Kirby, Robert W; Burrows, Jeremy N; Duffy, James; Peyton, David H; Reynolds, Kevin A; Kelly, Jane X; Kancharla, Papireddy; Buck, Alicia; Lee, Sohyon; Wegmann, Rebekka; Mena, Julien; Vasella, Flavio; Friesen, Julia; Regli, Luca; Le Rhun, Emilie; Zeitlberger, Anna Maria; Neidert, Marian Christoph; Tatari, Nazanin; Hutter, Gregor; Weller, Michael; Snijder, Berend; Weiss, Tobias

3-Position Biaryl Endochin-like Quinolones with Enhanced Antimalarial Performance

具有增强抗疟性能的3位联芳基内切辛类喹诺酮

Pou, Sovitj; Winter, Rolf W; Dodean, Rozalia A; Liebman, Katherine; Li, Yuexin; Mather, Michael W; Nepal, Binod; Nilsen, Aaron; Handford, Mason J; Riscoe, Teresa M; Laxson, Sydney; Kirtley, Payton J; Aleshnick, Maya; Zakharov, Lev N; Kelly, Jane X; Smilkstein, Martin J; Wilder, Brandon K; Kortagere, Sandhya; Vaidya, Akhil B; Alday, P Holland; Doggett, J Stone; Riscoe, Michael K

Synthesis of Deuterated Endochin-Like Quinolones

氘代内切辛类喹诺酮的合成

Pou, Sovitj; Winter, Rolf W; Liebman, Katherine M; Dodean, Rosie A; Nilsen, Aaron; DeBarber, Andrea; Doggett, J Stone; Riscoe, Michael K