Serendipitous and Systematic Chemoproteomic Discovery of MBLAC2, HINT1, and NME1-4 Inhibitors from Histone Deacetylase-Targeting Pharmacophores
从组蛋白去乙酰化酶靶向药效团中偶然发现和系统性化学蛋白质组学方法鉴定 MBLAC2、HINT1 和 NME1-4 抑制剂
期刊:ACS Chemical Biology
影响因子:3.8
doi:10.1021/acschembio.5c00108
Lechner, Severin; Sha, Shuyao; Sethiya, Jigar Paras; Szczupak, Patrycja; Dolot, Rafal; Lomada, Santosh; Sakhteman, Amirhossein; Tushaus, Johanna; Prokofeva, Polina; Krauss, Michael; Breu, Ferdinand; Vögerl, Katharina; Morgenstern, Martin; Hrabě de Angelis, Martin; Haucke, Volker; Wieland, Thomas; Wagner, Carston; Médard, Guillaume; Bracher, Franz; Kuster, Bernhard