日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CX-5461 Preferentially Induces Top2α-Dependent DNA Breaks at Ribosomal DNA Loci

CX-5461 优先诱导核糖体 DNA 位点的 Top2α 依赖性 DNA 断裂

Donald P Cameron, Jirawas Sornkom, Sameerh Alsahafi, Denis Drygin, Gretchen Poortinga, Grant A McArthur, Nadine Hein, Ross Hannan, Konstantin I Panov

Coinhibition of topoisomerase 1 and BRD4-mediated pause release selectively kills pancreatic cancer via readthrough transcription

拓扑异构酶1和BRD4介导的暂停释放的共同抑制可通过通读转录选择性地杀死胰腺癌细胞。

Donald P Cameron ,Jan Grosser ,Swetlana Ladigan ,Vladislav Kuzin ,Evanthia Iliopoulou ,Anika Wiegard ,Hajar Benredjem ,Kathryn Jackson ,Sven T Liffers ,Smiths Lueong ,Phyllis F Cheung ,Deepak Vangala ,Michael Pohl ,Richard Viebahn ,Christian Teschendorf ,Heiner Wolters ,Selami Usta ,Keyi Geng ,Claudia Kutter ,Marie Arsenian-Henriksson ,Jens T Siveke ,Andrea Tannapfel ,Wolff Schmiegel ,Stephan A Hahn ,Laura Baranello

MYC assembles and stimulates topoisomerases 1 and 2 in a "topoisome"

MYC 在“拓扑体”中组装并刺激拓扑异构酶 1 和 2。

Subhendu K Das ,Vladislav Kuzin ,Donald P Cameron ,Suzanne Sanford ,Rajiv Kumar Jha ,Zuqin Nie ,Marta Trullols Rosello ,Ronald Holewinski ,Thorkell Andresson ,Jan Wisniewski ,Toyoaki Natsume ,David H Price ,Brian A Lewis ,Fedor Kouzine ,David Levens ,Laura Baranello

MYCMI-7: A Small MYC-Binding Compound that Inhibits MYC: MAX Interaction and Tumor Growth in a MYC-Dependent Manner

MYCMI-7:一种小型 MYC 结合化合物,以 MYC 依赖的方式抑制 MYC:MAX 相互作用和肿瘤生长

Alina Castell, Qinzi Yan, Karin Fawkner, Wesam Bazzar, Fan Zhang, Malin Wickström, Mohammad Alzrigat, Marcela Franco, Cecilia Krona, Donald P Cameron, Cecilia Dyberg, Thale Kristin Olsen, Vasiliki Verschut, Linnéa Schmidt, Sheryl Y Lim, Loay Mahmoud, Per Hydbring, Sören Lehmann, Laura Baranello, Sve

TOP1 CAD-seq: A protocol to map catalytically engaged topoisomerase 1 in human cells

TOP1 CAD-seq:一种用于绘制人类细胞中催化活性拓扑异构酶1图谱的方案

Vladislav Kuzin,Anika Wiegard,Donald P Cameron,Laura Baranello

The Epstein-Barr virus deubiquitinating enzyme BPLF1 regulates the activity of topoisomerase II during productive infection

Epstein-Barr 病毒去泛素化酶 BPLF1 在生产性感染过程中调节拓扑异构酶 II 的活性

Jinlin Li, Noemi Nagy, Jiangnan Liu, Soham Gupta, Teresa Frisan, Thomas Hennig, Donald P Cameron, Laura Baranello, Maria G Masucci

Deficiency of Polη in Saccharomyces cerevisiae reveals the impact of transcription on damage-induced cohesion

酿酒酵母中 Polη 的缺乏揭示了转录对损伤诱导凝聚力的影响

Pei-Shang Wu, Jan Grosser, Donald P Cameron, Laura Baranello, Lena Ström

Changes in long-range rDNA-genomic interactions associate with altered RNA polymerase II gene programs during malignant transformation

长距离 rDNA-基因组相互作用的变化与恶性转化过程中 RNA 聚合酶 II 基因程序的改变有关

Jeannine Diesch, Megan J Bywater, Elaine Sanij, Donald P Cameron, William Schierding, Natalie Brajanovski, Jinbae Son, Jirawas Sornkom, Nadine Hein, Maurits Evers, Richard B Pearson, Grant A McArthur, Austen R D Ganley, Justin M O'Sullivan, Ross D Hannan, Gretchen Poortinga

Inhibition of Pol I transcription treats murine and human AML by targeting the leukemia-initiating cell population

抑制 Pol I 转录可通过靶向白血病起始细胞群来治疗小鼠和人类 AML

Nadine Hein, Donald P Cameron, Katherine M Hannan, Nhu-Y N Nguyen, Chun Yew Fong, Jirawas Sornkom, Meaghan Wall, Megan Pavy, Carleen Cullinane, Jeannine Diesch, Jennifer R Devlin, Amee J George, Elaine Sanij, Jaclyn Quin, Gretchen Poortinga, Inge Verbrugge, Adele Baker, Denis Drygin, Simon J Harriso

Inhibition of RNA polymerase I transcription initiation by CX-5461 activates non-canonical ATM/ATR signaling

CX-5461 抑制 RNA 聚合酶 I 转录起始可激活非典型 ATM/ATR 信号

Jaclyn Quin, Keefe T Chan, Jennifer R Devlin, Donald P Cameron, Jeannine Diesch, Carleen Cullinane, Jessica Ahern, Amit Khot, Nadine Hein, Amee J George, Katherine M Hannan, Gretchen Poortinga, Karen E Sheppard, Kum Kum Khanna, Ricky W Johnstone, Denis Drygin, Grant A McArthur, Richard B Pearson, El