Development of the First Low Nanomolar Liver Receptor Homolog-1 Agonist through Structure-guided Design.
通过结构导向设计开发首个低纳摩尔肝受体同源物-1激动剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.9b00753
Mays Suzanne G, Flynn Autumn R, Cornelison Jeffery L, Okafor C Denise, Wang Hongtao, Wang Guohui, Huang Xiangsheng, Donaldson Heather N, Millings Elizabeth J, Polavarapu Rohini, Moore David D, Calvert John W, Jui Nathan T, Ortlund Eric A