日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1H-indol-1-yl)benzenesulfonamide: A Novel Polypharmacology Agent to Target Carbonic Anhydrase IX and XII With Improved Selectivity, Wnt/β-Catenin Signaling Pathway, and P-Glycoprotein

4-(5-氯-3-(3,4,5-三甲氧基苯甲酰基)-1H-吲哚-1-基)苯磺酰胺:一种新型多靶点药物,可选择性地靶向碳酸酐酶IX和XII、Wnt/β-catenin信号通路以及P-糖蛋白。

Puxeddu, Michela; Bordone, Rosa; Colla, Claudia; Rotili, Gabriele; Coluccia, Antonio; Sciò, Pietro; Cuřínová, Petra; Nocentini, Alessio; Supuran, Claudiu T; Filiberti, Serena; Turati, Marta; Ronca, Roberto; Kopecka, Joanna; Riganti, Chiara; Jimenez, Lucia; Link, Wolfgang; Bigogno, Chiara; Dondio, Giulio; Barba, Martina; Canettieri, Gianluca; Silvestri, Romano; La Regina, Giuseppe

A global model-agnostic rule-based XAI method based on Parameterized Event Primitives for time series classifiers

一种基于参数化事件原语的全局模型无关的基于规则的XAI方法,用于时间序列分类器

Mekonnen, Ephrem Tibebe; Longo, Luca; Dondio, Pierpaolo

Novel N-(Heterocyclylphenyl)benzensulfonamide Sharing an Unreported Binding Site with T-Cell Factor 4 at the β-Catenin Armadillo Repeats Domain as an Anticancer Agent

新型N-(杂环苯基)苯磺酰胺与T细胞因子4在β-catenin Armadillo重复结构域共享一个未报道的结合位点,可作为抗癌剂

Marianna Nalli ,Laura Di Magno ,Yichao Wen ,Xin Liu ,Michele D'Ambrosio ,Michela Puxeddu ,Anastasia Parisi ,Jessica Sebastiani ,Andrea Sorato ,Antonio Coluccia ,Silvia Ripa ,Fiorella Di Pastena ,Davide Capelli ,Roberta Montanari ,Domiziana Masci ,Andrea Urbani ,Chiara Naro ,Claudio Sette ,Viviana Orlando ,Sara D'Angelo ,Stefano Biagioni ,Chiara Bigogno ,Giulio Dondio ,Arianna Pastore ,Mariano Stornaiuolo ,Gianluca Canettieri ,Te Liu ,Romano Silvestri ,Giuseppe La Regina

Favorable Preclinical Pharmacological Profile of a Novel Antimalarial Pyrrolizidinylmethyl Derivative of 4-amino-7-chloroquinoline with Potent In Vitro and In Vivo Activities

一种新型抗疟吡咯里西啶甲基衍生物(4-氨基-7-氯喹啉)具有良好的临床前药理学特性,并表现出强大的体外和体内活性。

Basilico, Nicoletta; Parapini, Silvia; D'Alessandro, Sarah; Misiano, Paola; Romeo, Sergio; Dondio, Giulio; Yardley, Vanessa; Vivas, Livia; Nasser, Shereen; Rénia, Laurent; Russell, Bruce M; Suwanarusk, Rossarin; Nosten, François; Sparatore, Anna; Taramelli, Donatella

Survey data on dysfunctional attitudes, personality traits, and agreement with persuasive techniques

关于不良态度、人格特质以及对说服技巧认同度的调查数据

Braca, Annye; Dondio, Pierpaolo

Discovery of RC-752, a Novel Sigma-1 Receptor Antagonist with Antinociceptive Activity: A Promising Tool for Fighting Neuropathic Pain

发现具有抗伤害活性的新型 Sigma-1 受体拮抗剂 RC-752:一种有前途的抗击神经性疼痛的工具

Giacomo Rossino, Annamaria Marra, Roberta Listro, Marco Peviani, Elena Poggio, Daniela Curti, Giorgia Pellavio, Umberto Laforenza, Giulio Dondio, Dirk Schepmann, Bernhard Wünsch, Martina Bedeschi, Noemi Marino, Anna Tesei, Hee-Jin Ha, Young-Ho Kim, Jihyae Ann, Jeewoo Lee, Pasquale Linciano, Marcello

Induction of Ferroptosis in Glioblastoma and Ovarian Cancers by a New Pyrrole Tubulin Assembly Inhibitor

新型吡咯微管蛋白组装抑制剂诱导胶质母细胞瘤和卵巢癌中的铁死亡

Michela Puxeddu, Jianchao Wu, Ruoli Bai, Michele D'Ambrosio, Marianna Nalli, Antonio Coluccia, Simone Manetto, Alessia Ciogli, Domiziana Masci, Andrea Urbani, Cinzia Fionda, Sonia Coni, Rosa Bordone, Gianluca Canettieri, Chiara Bigogno, Giulio Dondio, Ernest Hamel, Te Liu, Romano Silvestri, Giuseppe

Givinostat-Liposomes: Anti-Tumor Effect on 2D and 3D Glioblastoma Models and Pharmacokinetics

Givinostat-脂质体:对 2D 和 3D 胶质母细胞瘤模型的抗肿瘤作用和药代动力学

Lorenzo Taiarol, Chiara Bigogno, Silvia Sesana, Marcelo Kravicz, Francesca Viale, Eleonora Pozzi, Laura Monza, Valentina Alda Carozzi, Cristina Meregalli, Silvia Valtorta, Rosa Maria Moresco, Marcus Koch, Federica Barbugian, Laura Russo, Giulio Dondio, Christian Steinkühler, Francesca Re

Discovery of Reversible Inhibitors of KDM1A Efficacious in Acute Myeloid Leukemia Models

发现对急性髓系白血病模型有效的KDM1A可逆抑制剂

Romussi, Alessia; Cappa, Anna; Vianello, Paola; Brambillasca, Silvia; Cera, Maria Rosaria; Dal Zuffo, Roberto; Fagà, Giovanni; Fattori, Raimondo; Moretti, Loris; Trifirò, Paolo; Villa, Manuela; Vultaggio, Stefania; Cecatiello, Valentina; Pasqualato, Sebastiano; Dondio, Giulio; So, Chi Wai Eric; Minucci, Saverio; Sartori, Luca; Varasi, Mario; Mercurio, Ciro

Anti-tumor Efficacy Assessment of the Sigma Receptor Pan Modulator RC-106. A Promising Therapeutic Tool for Pancreatic Cancer

Sigma受体泛调节剂RC-106的抗肿瘤疗效评估:一种有前景的胰腺癌治疗工具

Tesei, Anna; Cortesi, Michela; Pignatta, Sara; Arienti, Chiara; Dondio, Giulio Massimo; Bigogno, Chiara; Malacrida, Alessio; Miloso, Mariarosaria; Meregalli, Cristina; Chiorazzi, Alessia; Carozzi, Valentina; Cavaletti, Guido; Rui, Marta; Marra, Annamaria; Rossi, Daniela; Collina, Simona