日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cooperativity and communication between the active sites of the dimeric SARS-CoV-2 main protease

二聚体SARS-CoV-2主蛋白酶活性位点之间的协同作用和通讯

Zvornicanin, Sarah N; Shaqra, Ala M; Flynn, Julia; Intravaia, Lauren E; Martinez, Heidi Carias; Jia, Weiping; Gupta, Devendra Kumar; Moquin, Stephanie; Dovala, Dustin; Bolon, Daniel N; Kelch, Brian A; Schiffer, Celia A; Yilmaz, Nese Kurt

Discovery of EGT710, an Oral Nonpeptidomimetic Reversible Covalent SARS-CoV-2 Main Protease Inhibitor

发现 EGT710,一种口服非肽模拟可逆共价 SARS-CoV-2 主蛋白酶抑制剂

Papillon, Julien P N; Yuan, Jun; Hesse, Matthew J; Zhang, Lei; Robinson, Richard I; Ware, Nathaniel F; Hornak, Viktor; Karki, Rajeshri G; Kirrane, Tom; Garland, Keira; Joseph, Sajan; Moquin, Stephanie A; Lakshminarayana, Suresh B; Tandeske, Laura; Dovala, Dustin; Knapp, Mark; Ornelas, Elizabeth; Fuller, Daniel; Ho, Pei-I; Xie, Xuping; Vulic, Katarina; Skolnik, Suzanne M; Gao, Jinhai; Zambrowski, Mark; Spiess, Meike; Duca, José S; Busby, Scott A; Schirle, Markus; Robinson, Michael; Shi, Pei-Yong; Moser, Heinz E; Sarko, Christopher; Bradner, James E; Diagana, Thierry T; Tallarico, John A

Molecular mechanisms of drug resistance and compensation in SARS-CoV-2 main protease: the interplay between E166 and L50

SARS-CoV-2 主蛋白酶的耐药性和补偿的分子机制:E166 和 L50 之间的相互作用

Zvornicanin, Sarah N; Shaqra, Ala M; Flynn, Julia; Carias Martinez, Heidi; Jia, Weiping; Moquin, Stephanie; Dovala, Dustin; Bolon, Daniel N; Kurt Yilmaz, Nese; Schiffer, Celia A

Structural Analysis of Inhibitor Binding to the Feline Enteric Coronavirus (FECV) Main Protease

抑制剂与猫肠道冠状病毒(FECV)主蛋白酶结合的结构分析

Maryam, Arooma; Moquin, Stephanie A; Dovala, Dustin; Kaur, Jagroop; Kurt Yilmaz, Nese; Shaqra, Ala M; Schiffer, Celia A

Targeted Transcriptional Repression by Induced Proximity

诱导邻近效应介导的靶向转录抑制

Stieger, Christian E; Chen, Xinru; Dovala, Dustin; Wu, Fabian; Pizzato, Nicolas; McKenna, Jeffrey; Johannessen, Cory; Fodor, Barna D; Schirle, Markus; Nomura, Daniel K

Sulfinyl Aziridines as Stereoselective Covalent Destabilizing Degraders of the Oncogenic Transcription Factor MYC.

亚磺酰基氮丙啶作为致癌转录因子MYC的立体选择性共价去稳定化降解剂

Rosen Hannah T, Li Kelvin, Li Erin L, Currier Brynne, Brittain Scott M, Garcia Francisco J, Beard Diana C, Haenni-Holzinger Sandra, Dovala Dustin, McKenna Jeffrey M, Schirle Markus, Maimone Thomas J, Nomura Daniel K

Rational Chemical Design of Molecular Glue Degraders

分子胶降解剂的合理化学设计

Toriki, Ethan S; Papatzimas, James W; Nishikawa, Kaila; Dovala, Dustin; Frank, Andreas O; Hesse, Matthew J; Dankova, Daniela; Song, Jae-Geun; Bruce-Smythe, Megan; Struble, Heidi; Garcia, Francisco J; Brittain, Scott M; Kile, Andrew C; McGregor, Lynn M; McKenna, Jeffrey M; Tallarico, John A; Schirle, Markus; Nomura, Daniel K

Correction to "Rational Chemical Design of Molecular Glue Degraders"

对“分子胶降解剂的合理化学设计”的更正

Toriki, Ethan S; Papatzimas, James W; Nishikawa, Kaila; Dovala, Dustin; Frank, Andreas O; Hesse, Matthew J; Dankova, Daniela; Song, Jae-Geun; Bruce-Smythe, Megan; Struble, Heidi; Garcia, Francisco J; Brittain, Scott M; Kile, Andrew C; McGregor, Lynn M; McKenna, Jeffrey M; Tallarico, John A; Schirle, Markus; Nomura, Daniel K

Crystal Structures of Inhibitor-Bound Main Protease from Delta- and Gamma-Coronaviruses

δ冠状病毒和γ冠状病毒抑制剂结合主蛋白酶的晶体结构

Zvornicanin, Sarah N; Shaqra, Ala M; Huang, Qiuyu J; Ornelas, Elizabeth; Moghe, Mallika; Knapp, Mark; Moquin, Stephanie; Dovala, Dustin; Schiffer, Celia A; Kurt Yilmaz, Nese

De novo Design of SARS-CoV-2 Main Protease Inhibitors

SARS-CoV-2 主蛋白酶抑制剂的全新设计

Fischer, Christian; Vepřek, Nynke A; Peitsinis, Zisis; Rühmann, Klaus-Peter; Yang, Chao; Spradlin, Jessica N; Dovala, Dustin; Nomura, Daniel K; Zhang, Yingkai; Trauner, Dirk