Use of protease substrate specificity screening in the rational design of selective protease inhibitors with unnatural amino acids: Application to HGFA, matriptase, and hepsin.
利用蛋白酶底物特异性筛选合理设计含非天然氨基酸的选择性蛋白酶抑制剂:应用于 HGFA、matriptase 和 hepsin
期刊:Protein Science
影响因子:5.2
doi:10.1002/pro.5110
Mahoney Matthew W, Helander Jonathan, Kooner Anoopjit S, Norman Mariah, Damalanka Vishnu C, De Bona Paolo, Kasperkiewicz Paulina, Rut Wioletta, Poreba Marcin, Kashipathy Maithri M, Battaile Kevin P, Lovell Scott, O'Donoghue Anthony J, Craik Charles S, Drag Marcin, Janetka James W