日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Self-Masked Aldehyde Inhibitors: A Novel Strategy for Inhibiting Cysteine Proteases

自掩蔽醛抑制剂:抑制半胱氨酸蛋白酶的新策略

Linfeng Li, Bala C Chenna, Kai S Yang, Taylor R Cole, Zachary T Goodall, Miriam Giardini, Zahra Moghadamchargari, Elizabeth A Hernandez, Jana Gomez, Claudia M Calvet, Jean A Bernatchez, Drake M Mellott, Jiyun Zhu, Andrew Rademacher, Diane Thomas, Lauren R Blankenship, Aleksandra Drelich, Arthur Laga

Bepridil is potent against SARS-CoV-2 in vitro

贝普地尔在体外对 SARS-CoV-2 有疗效

Erol C Vatansever, Kai S Yang, Aleksandra K Drelich, Kaci C Kratch, Chia-Chuan Cho, Kempaiah Rayavara Kempaiah, Jason C Hsu, Drake M Mellott, Shiqing Xu, Chien-Te K Tseng, Wenshe Ray Liu

Peptidomimetic Vinyl Heterocyclic Inhibitors of Cruzain Effect Antitrypanosomal Activity

肽模拟乙烯基杂环抑制剂 Cruzain 效应抗锥虫活性

Bala C Chenna, Linfeng Li, Drake M Mellott, Xiang Zhai, Jair L Siqueira-Neto, Claudia Calvet Alvarez, Jean A Bernatchez, Emily Desormeaux, Elizabeth Alvarez Hernandez, Jana Gomez, James H McKerrow, Jorge Cruz-Reyes, Thomas D Meek

Bepridil is potent against SARS-CoV-2 In Vitro

贝普地尔在体外对 SARS-CoV-2 有疗效

Erol C Vatansever, Kai Yang, Kaci C Kratch, Aleksandra Drelich, Chia-Chuan Cho, Drake M Mellott, Shiqing Xu, Chien-Te K Tseng, Wenshe Ray Liu

A cysteine protease inhibitor blocks SARS-CoV-2 infection of human and monkey cells

半胱氨酸蛋白酶抑制剂可阻断 SARS-CoV-2 感染人类和猴细胞

Drake M Mellott, Chien-Te Tseng, Aleksandra Drelich, Pavla Fajtová, Bala C Chenna, Demetrios H Kostomiris, Jason Hsu, Jiyun Zhu, Zane W Taylor, Vivian Tat, Ardala Katzfuss, Linfeng Li, Miriam A Giardini, Danielle Skinner, Ken Hirata, Sungjun Beck, Aaron F Carlin, Alex E Clark, Laura Beretta, Daniel