日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A fission yeast-based platform for nematode PDE inhibitor discovery

基于裂殖酵母的线虫PDE抑制剂发现平台

Bibeau, Sarah; Chen, Natalie; Sutoris, Hannah; Ly, Judy; Eberhard, Jeremy; Hubbell, Sara M; Banda, Eric; Povh, Esther; Anindya, Clianta S; Berwanger, Michael R; Sinise, Sarah E; Zhang, Xieyang; Morken, James P; Galande, Kranti K; Cote, Rick H; Dranchak, Patricia K; Inglese, James; Hoffman, Charles S

A general assay platform to study protein pharmacology using ligand-dependent structural dynamics.

利用配体依赖性结构动力学研究蛋白质药理学的通用检测平台

Ciulla Daniel A, Dranchak Patricia K, Aitha Mahesh, van Neer Renier H P, Shah Divia, Tharakan Ravi, Wilson Kelli M, Wang Yuhong, Braisted John C, Inglese James

Metabolic engineering and late-stage functionalization expand the chemical space of the antimalarial premarineosin A

代谢工程和后期功能化扩展了抗疟药普瑞马利尼奥辛A的化学空间。

McBride, Christina M; McCauley, Morgan; Harris, Natalia R; Amin, Sahar; Curtis, Brian J; Verhey-Henke, Linnea; Teklemichael, Awet A; Oliphant, Erin N; Dranchak, Patricia; Lev, Katherine L; Qu, Fengrui; Snodgrass, Harrison M; Lewis, Jared C; Inglese, James; Su, Xin-Zhuan; Pereira, Filipa; Sherman, David H

A Quantitative High-Throughput Screen Identifies Compounds that Upregulate the p53 Isoform Δ133p53α and Inhibit Cellular Senescence.

定量高通量筛选鉴定出能上调 p53 同工型 Δ133p53α 并抑制细胞衰老的化合物

Lissa Delphine, Joruiz Sebastien M, Dranchak Patricia K, Ungerleider Kyra, Yamada Leo, Horikawa Izumi, Oliphant Erin, Manubag Rebecca, Von Muhlinen Natalia, Beck Jessica, Harris Brent T, Inglese James, Harris Curtis

Pharmacologic activation of Δ133p53α reduces cellular senescence in progeria patients-derived cells

药物激活Δ133p53α可减少早衰症患者来源细胞的衰老

Joruiz, Sebastien M; Lissa, Delphine; Von Muhlinen, Natalia; Dranchak, Patricia K; Inglese, James; Horikawa, Izumi; Harris, Curtis C

Methotrexate-based PROTACs as DHFR-specific chemical probes

基于甲氨蝶呤的 PROTAC 作为 DHFR 特异性化学探针

Sandeep Rana, Patricia Dranchak, Jayme L Dahlin, Laurence Lamy, Wenqing Li, Erin Oliphant, Jonathan H Shrimp, Girish H Rajacharya, Ravi Tharakan, David O Holland, Apryl S Whitten, Kelli M Wilson, Pankaj K Singh, Scott K Durum, Dingyin Tao, Ganesha Rai, James Inglese

Machine Learning Models Identify Inhibitors of New Delhi Metallo-β-lactamase

机器学习模型识别新德里金属-β-内酰胺酶抑制剂

Zishuo Cheng, Mahesh Aitha, Caitlyn A Thomas, Aidan Sturgill, Mitch Fairweather, Amy Hu, Christopher R Bethel, Dann D Rivera, Patricia Dranchak, Pei W Thomas, Han Li, Qi Feng, Kaicheng Tao, Minshuai Song, Na Sun, Shuo Wang, Surendra Bikram Silwal, Richard C Page, Walt Fast, Robert A Bonomo, Maria We

A Differential Ion Mobility Acoustic Ejection Mass Spectrometer System for Screening Isomerization-Mediating Enzyme Drug Targets

用于筛选异构化介导酶药物靶点的差分离子迁移率声波喷射质谱仪系统

Bazargan, Samad; Dranchak, Patricia; Liu, Chang; Inglese, James; Janiszewski, John; Schneider, Bradley B; Covey, Thomas R

In vivo quantitative high-throughput screening for drug discovery and comparative toxicology

用于药物发现和比较毒理学的体内定量高通量筛选

Patricia K Dranchak, Erin Oliphant, Bryan Queme, Laurence Lamy, Yuhong Wang, Ruili Huang, Menghang Xia, Dingyin Tao, James Inglese

High-throughput screening identifies cell cycle-associated signaling cascades that regulate a multienzyme glucosome assembly in human cells

高通量筛选鉴定出调节人类细胞中多酶葡萄糖体组装的细胞周期相关信号级联

Danielle L Schmitt, Patricia Dranchak, Prakash Parajuli, Dvir Blivis, Ty Voss, Casey L Kohnhorst, Minjoung Kyoung, James Inglese, Songon An