日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of an ITK and TRK kinase inhibitor for the potential topical treatment of atopic dermatitis

发现一种ITK和TRK激酶抑制剂,可用于治疗特应性皮炎。

Duffen, Jennifer L; Crouse, Kimberly K; Ji, Lin; Brault, Amy L; Ford, Kristen; Brooks, Jonathan; Jelinsky, Scott A; Li, Yizheng; Shin, Julia H; Zhao, Yajuan; Andreyeva, Tatyana; Hammerman, Katherine; Arnold, Christina; Sheldon, Richard T; Garren, Jeonifer; LaBarge, Wes; Resek, Anthony; Volmer, Jon; Bagley, Scott W; Casimiro-Garcia, Agustin; Chinigo, Gary M; Davoren, Jennifer E; Denny, Rajiah Aldrin; Drozda, Susan; Foley, Timothy L; Hicklin, Robert W; Liu, Shenping; Lovering, Frank E; Nedoma, Nicole L; Parikh, Mihir D; Strohbach, Joseph W; Trujillo, John I; Steyn, Stefanus J; Nocka, Karl; Hegen, Martin; Vincent, Fabien; Lee, Katherine L; Gerstenberger, Brian S; Primiano, Michael J

Inhibiting peptidylarginine deiminases (PAD1-4) by targeting a Ca(2+) dependent allosteric binding site.

通过靶向 Ca(2+) 依赖性变构结合位点来抑制肽基精氨酸脱亚胺酶 (PAD1-4)

Dakin Leslie A, Xing Li, Hall Justin, Ding Weidong, Vajdos Felix F, Pelker Jeffrey W, Ramsey Simeon, Balbo Paul, Sahasrabudhe Parag V, Banker Mary Ellen, Choi Won Young, Wright Stephen W, Chang Jeanne S, Curto John M, Davoren Jennifer E, Drozda Susan E, Fennell Kimberly F, Futatsugi Kentaro, Kortum Steve, Lee Katherine L, Liu Shenping, Lovering Frank, Nicki Jennifer A, Trujillo John I, Vincent Fabien, Schnute Mark E

Peptidylarginine Deiminase (PAD) Inhibitor Optimization through Displacement of a Trapped Water Molecule

通过置换被捕获的水分子来优化肽基精氨酸脱亚胺酶(PAD)抑制剂

Schnute, Mark E; Chinigo, Gary M; Futatsugi, Kentaro; Yamaguchi, Masaya; Bagley, Scott W; Banker, Mary Ellen; Chang, Jeanne S; Chen, Ming Z; Choi, Won Young; Corbett, Matthew S; Drozda, Susan E; Ebner, David C; Garcia-Irizarry, Carmen; Hicklin, Robert; Hoy, Susan; Jiao, Wenhua; Kortum, Steven; Lee, Katherine L; Limburg, David C; Lovering, Frank; Moreno, Antonio; Mousseau, James J; Pan, Senliang; Parikh, Mihir D; Pelker, Jeffrey W; Ramsey, Simeon; Reilly, Usa; Rescourio, Gwenaella; Schmitt, Daniel C; Simpson, Brittany; Skrzypek, Grzegorz J; Smaltz, Daniel J; Taylor, Alexandria P; Torella, Rubben; Trujillo, John I; Vajdos, Felix F; Wepy, James A; Wright, Stephen W; Blakemore, David C; Vincent, Fabien; Clerin, Valerie M

Toxoplasma FER1 is a versatile and dynamic mediator of differential microneme trafficking and microneme exocytosis

弓形虫 FER1 是一种多功能且动态的微粒体运输和微粒体胞吐介质。

Tagoe, Daniel N A; Ribeiro E Silva, Adeline; Drozda, Allison A; Coppens, Isabelle; Coleman, Bradley I; Gubbels, Marc-Jan

Integrating real-world data to assess cardiac ablation device outcomes in a multicenter study using the OMOP common data model for regulatory decisions: implementation and evaluation

利用OMOP通用数据模型,在多中心研究中整合真实世界数据以评估心脏消融装置的疗效,从而为监管决策提供依据:实施与评估

Yu, Yue; Jiang, Guoqian; Brandt, Eric; Forsyth, Tom; Dhruva, Sanket S; Zhang, Shumin; Chen, Jiajing; Noseworthy, Peter A; Doshi, Amit A; Collison-Farr, Kimberly; Kim, Dure; Ross, Joseph S; Coplan, Paul M; Drozda, Joseph P Jr

Ancient retroperitoneal schwannoma imitating seminoma recurrence: A case report

一例疑似精原细胞瘤复发的古老型腹膜后神经鞘瘤:病例报告

Horak, Samuel; Cierna, Zuzana; Kopecka, Iveta; Drozda, Vladimir; Harmanos, Michal; Cvik, Marian

Safety and Effectiveness of a Catheter With Contact Force and 6-Hole Irrigation for Ablation of Persistent Atrial Fibrillation in Routine Clinical Practice

在常规临床实践中,采用接触力和六孔灌注导管消融治疗持续性房颤的安全性和有效性

Dhruva, Sanket S; Zhang, Shumin; Chen, Jiajing; Noseworthy, Peter A; Doshi, Amit A; Agboola, Kolade M; Herrin, Jeph; Jiang, Guoqian; Yu, Yue; Cafri, Guy; Collison Farr, Kimberly; Ervin, Keondae R; Ross, Joseph S; Coplan, Paul M; Drozda, Joseph P Jr

Targeting carbonic anhydrase IX and XII isoforms with small molecule inhibitors and monoclonal antibodies

利用小分子抑制剂和单克隆抗体靶向碳酸酐酶IX和XII同工酶

Kciuk, Mateusz; Gielecińska, Adrianna; Mujwar, Somdutt; Mojzych, Mariusz; Marciniak, Beata; Drozda, Rafał; Kontek, Renata

Insights into the expression of DNA (de)methylation genes responsive to nitric oxide signaling in potato resistance to late blight disease

深入了解响应一氧化氮信号传导的DNA(去)甲基化基因在马铃薯晚疫病抗性中的表达

Drozda, Andżelika; Kurpisz, Barbara; Guan, Yufeng; Arasimowicz-Jelonek, Magdalena; Plich, Jarosław; Jagodzik, Przemysław; Kuźnicki, Daniel; Floryszak-Wieczorek, Jolanta

Multi-institutional distributed data networks for real-world evidence about medical devices: building unique device identifiers into longitudinal data (BUILD)

用于获取医疗器械真实世界证据的多机构分布式数据网络:将唯一设备标识符构建到纵向数据中(BUILD)

Drozda, Joseph P Jr; Graham, Jove; Muhlestein, Joseph B; Tcheng, James E; Roach, James; Forsyth, Tom; Knight, Stacey; McKinnon, Andrew; May, Heidi; Wilson, Natalia A; Berlin, Jesse A; Simard, Edgar P