日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development and characterization of endolysosomal trafficking targeting chimera degraders of α(1A)-adrenergic receptor.

开发和表征靶向α(1A)-肾上腺素能受体嵌合降解剂的内溶酶体运输。

Chen Jiwei, Wang Shuo, Li Tong, Li Wenhua, Ke Xuechun, Ma Zhao, Du Lupei, Li Minyong

Erratum: Author correction to "Identification of anthelmintic parbendazole as a therapeutic molecule for HNSCC through connectivity map-based drug repositioning" [Acta Pharm Sin B 12 (2022) 2429-2442]

勘误:作者对“通过基于连接图的药物重定位鉴定抗蠕虫药帕苯达唑作为头颈部鳞状细胞癌的治疗分子”[Acta Pharm Sin B 12 (2022) 2429-2442]进行了更正。

Liang, Dong; Yu, Chen; Ma, Zhao; Yang, Xingye; Li, Zhenzhen; Dong, Xuhui; Qin, Xiaojun; Du, Lupei; Li, Minyong

Deuteration-Driven Photopharmacology: Deuterium-Labeled AzoCholine for Controlling Alpha 7 Nicotinic Acetylcholine Receptors

氘代驱动的光药理学:氘标记的偶氮胆碱用于控制α7尼古丁乙酰胆碱受体

Yang, Xingye; Zhou, Xin; Qin, Xiaojun; Liang, Dong; Dong, Xuhui; Ji, Huimin; Wen, Siman; Du, Lupei; Li, Minyong

Novel BRD4-p53 Inhibitor SDU-071 Suppresses Proliferation and Migration of MDA-MB-231 Triple-Negative Breast Cancer Cells.

新型 BRD4-p53 抑制剂 SDU-071 可抑制 MDA-MB-231 三阴性乳腺癌细胞的增殖和迁移

Wang Shumei, Lei Kang, Lai Hsien-Tsung, Liu Tingting, Du Lupei, Wu Shwu-Yuan, Ye Xiaohan, Chiang Cheng-Ming, Li Minyong

Fluorescent Ligand-Based Discovery of Small-Molecule Sulfonamide Agonists for GPR120

基于荧光配体的小分子磺酰胺类GPR120激动剂的发现

Ma, Siyue; Li, Zhenzhen; Yang, Yueli; Zhang, Ling; Li, Minyong; Du, Lupei

Visualization-Based Discovery of Vanin-1 Inhibitors for Colitis

基于可视化的Vanin-1抑制剂在结肠炎治疗中的发现

Wang, Guankai; Wang, Jingjing; Du, Lupei; Li, Minyong

Polarity-based fluorescence probes: properties and applications

基于极性的荧光探针:性质和应用

Qin, Xiaojun; Yang, Xingye; Du, Lupei; Li, Minyong

Aggregation-Induced Emission: Lighting Up hERG Potassium Channel

聚集诱导发光:激活 hERG 钾通道

Zhang, Xiaomeng; Liu, Tingting; Li, Qi; Li, Minyong; Du, Lupei

Astemizole-based turn-on fluorescent probes for imaging hERG potassium channel

基于阿司咪唑的开启型荧光探针用于hERG钾通道成像

Zhang, Xiaomeng; Liu, Tingting; Wang, Beilei; Gao, Yuqi; Liu, Pan; Li, Minyong; Du, Lupei

Environment-sensitive turn-on fluorescent probes for p53-MDM2 protein-protein interaction

用于检测p53-MDM2蛋白-蛋白相互作用的环境敏感型荧光探针

Liu, Tingting; Jiang, Yan; Liu, Zhenzhen; Li, Jin; Fang, Kun; Zhuang, Chunlin; Du, Lupei; Fang, Hao; Sheng, Chunquan; Li, Minyong