Discovery of a "First-in-Class" Selective Multikinase (CDK4/6/9-AURKA/B) Inhibitor, LCI133, for Neuroblastoma
发现一种“首创”的选择性多激酶(CDK4/6/9-AURKA/B)抑制剂LCI133,用于治疗神经母细胞瘤
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c01688
Maddeboina, Krishnaiah; Pal, Dhananjaya; Yada, Bharath; McHale, Cody C; Singh, Sandeep K; Chhonker, Yashpal S; Dryden, Hailey L; Delara, Ritchie; Mujumdar, Vaidehi; Zhang, Qi; Murry, Daryl J; Durden, Donald L