日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Excelsatoxin A-Receptor TMEM233 Modulates Nav1.8

Excelsatoxin A 受体 TMEM233 调节 Nav1.8

Oprita, George; Meyer, Marvin J A; Rudolf, Daniel; Pombeiro Stein, Inês C A; Deuis, Jennifer R; Tran, Hue N T; Durek, Thomas; Tabea, Klasfauseweh; Sina, Jami; Waxman, Stephen G; Dib-Hajj, Sulayman D; Babes, Alexandru; Vetter, Irina; Leffler, Andreas

Enzyme-Assisted Synthesis and In Vitro Characterization of Bifunctional PCSK9 Inhibitors.

酶辅助合成双功能PCSK9抑制剂及其体外表征。

Zhang Yuhui, Wang Li, Corcilius Leo, Reji Amal K, Payne Richard J, Hong Bin, Durek Thomas, Wang Conan K, Craik David J

Asparaginyl Ligases with Engineered Substrate Specificity for Controlled, Sequential Transpeptidation Reactions

具有工程化底物特异性的天冬酰胺连接酶用于可控的、顺序的转肽反应

Zhou, Yan; de Veer, Simon J; Tyler, Tristan J; Chen, Yufei; Durek, Thomas; Craik, David J; Rehm, Fabian B H

Yeast as a tool for exploring disulfide-rich peptides

利用酵母作为探索富含二硫键肽的工具

Yap, Kuok; Porth, Owen T; Xie, Jing; Wang, Conan K; Durek, Thomas; Wittrup, K Dane; Craik, David J

Cyclization of the Analgesic α-Conotoxin Vc1.1 With a Non-Natural Linker: Effects on Structure, Stability, and Bioactivity

利用非天然连接基环化镇痛剂α-芋螺毒素Vc1.1:对结构、稳定性和生物活性的影响

Zhang, Yuhui; Tae, Han Shen; Adams, David J; Durek, Thomas; Craik, David J

Repurposing a plant peptide cyclase for targeted lysine acylation

利用植物肽环化酶进行靶向赖氨酸酰化

Rehm, Fabian B H; Tyler, Tristan J; Zhou, Yan; Huang, Yen-Hua; Wang, Conan K; Lawrence, Nicole; Craik, David J; Durek, Thomas

Author Correction: Repurposing a plant peptide cyclase for targeted lysine acylation

作者更正:植物肽环化酶的再利用及其在靶向赖氨酸酰化中的应用

Rehm, Fabian B H; Tyler, Tristan J; Zhou, Yan; Huang, Yen-Hua; Wang, Conan K; Lawrence, Nicole; Craik, David J; Durek, Thomas

Tertiary amide bond formation by an engineered asparaginyl ligase

利用工程改造的天冬酰胺连接酶形成叔酰胺键

de Veer, Simon J; Zhou, Yan; Durek, Thomas; Craik, David J; Rehm, Fabian B H

Revealing molecular determinants governing mambalgin-3 pharmacology at acid-sensing ion channel 1 variants

揭示酸敏感离子通道 1 变体中 mambalgin-3 药理学的分子决定因素

Cristofori-Armstrong, Ben; Budusan, Elena; Smith, Jennifer J; Reynaud, Steve; Voll, Kerstin; Chassagnon, Irène R; Durek, Thomas; Rash, Lachlan D

Nucleation of a key beta-turn promotes cyclotide oxidative folding

关键β-转角的成核促进环肽的氧化折叠

Tian, Sixin; de Veer, Simon J; Durek, Thomas; Wang, Conan K; Craik, David J