日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting replication stress in neuroblastoma by exploiting the synergistic potential of second generation RRM2 and CHK1 inhibitors

利用第二代RRM2和CHK1抑制剂的协同作用,靶向治疗神经母细胞瘤中的复制应激

Nelen, Iris H; Leys, Soetkin; Bekaert, Sarah-Lee; De Vloed, Fanny; Martens, Fien; Sanders, Ellen; Praveena Enton Raj, Angeline; Jeschke, Annika; Ohmura, Shunya; Grünewald, Thomas G P; Mus, Liselot M; Lammens, Tim; Van Roy, Nadine; De Wilde, Bram; Speleman, Frank; Van Hemelryk, Annelies; Depestel, Lisa; Durinck, Kaat

Pathway for the Development of ATR Inhibitors in Pediatric Malignancies: An ACCELERATE Multistakeholder Analysis

儿童恶性肿瘤中ATR抑制剂的研发路径:一项ACCELERATE多方利益相关者分析

Gatz, Susanne A; Glade-Bender, Julia; Pearson, Andrew D J; Ortiz, Michael V; Bernardi, Ronald; Chesler, Lou; Clifford, Steve; Cohen-Gogo, Sarah; De La Cuesta, Esther; de Rojas, Teresa; Durinck, Kaat; Federico, Sara; Fox, Elizabeth; George, Sally; Gounaris, Ioannis; Henssen, Anton George; Irwin, Meredith; Kool, Marcel; Lau, Alan; Nysom, Karsten; Pappo, Alberto; Pennock, Gregory K; Pfister, Stefan M; Scobie, Nicole; Slotkin, Emily K; Smith, Malcolm; Speleman, Frank; Stewart, Elizabeth A; Weigel, Brenda J; Vassal, Gilles

RUVBL1 and RUVBL2 are druggable MYC effector regulators in neuroblastoma cells

RUVBL1 和 RUVBL2 是神经母细胞瘤细胞中可作为药物靶点的 MYC 效应调节因子。

Siaw, Joachim Tetteh; Claeys, Arne; Lai, Wei-Yun; Borenäs, Marcus; Hilgert, Elien; Bekaert, Sarah-Lee; Sanders, Ellen; Kaya, Irem; Van Dorpe, Jo; Speleman, Frank; Durinck, Kaat; Hallberg, Bengt; Palmer, Ruth H; Van den Eynden, Jimmy

Second-Generation AURKA-Targeting PROTACs: Structural Optimization toward in Vivo Degradation in Neuroblastoma

第二代靶向AURKA的PROTAC:针对神经母细胞瘤体内降解的结构优化

Krols, Simon; Rishfi, Muhammad; Martens, Fien; Van Hauwermeiren, Anouk; Sanders, Ellen; De Sutter, Pieter-Jan; Vermeulen, An; De Wever, Kaat; Bekaert, Sarah-Lee; Dolman, M Emmy M; Tax, Gabor; Kamili, Alvin; Fletcher, Jamie I; Depestel, Lisa; De Wilde, Bram; Durinck, Kaat; Van Calenbergh, Serge

Synergistic inhibition of CHK1 and MUS81 to combat replication stress resistance in high-risk neuroblastoma.

协同抑制 CHK1 和 MUS81 以对抗高危神经母细胞瘤的复制应激抵抗。

Hilgert Elien, Van Neste Christophe, Bekaert Sarah-Lee, Martens Fien, Vanhauwaert Suzanne, Sanders Ellen, Verstraelen Peter, Risseeuw Martijn, Westerhout Ellen M, Grannetia Mark A, Van Calenbergh Serge, Van Roy Nadine, De Vos Winnok H, Wolthuis Rob W F, Speleman Frank, Depestel Lisa, Durinck Kaat

Induction of a distinct macrophage population and protection from lung injury and fibrosis by Notch2 blockade.

Notch2阻断可诱导产生独特的巨噬细胞群,并保护肺部免受损伤和纤维化

Cruz Tleugabulova Mayra, Melo Sandra P, Wong Aaron, Arlantico Alexander, Liu Meizi, Webster Joshua D, Lau Julia, Lechner Antonie, Corak Basak, Hodgins Jonathan J, Garlapati Venkata S, De Simone Marco, Korin Ben, Avraham Shimrit, Lund Jessica, Jeet Surinder, Reiss Alexander, Bender Hannah, Austin Cary D, Darmanis Spyros, Modrusan Zora, Brightbill Hans, Durinck Steffen, Diamond Michael S, Schneider Christoph, Shaw Andrey S, Nitschké Maximilian

Comparative genomics incorporating translocation renal cell carcinoma mouse model reveals molecular mechanisms of tumorigenesis

结合易位性肾细胞癌小鼠模型的比较基因组学揭示了肿瘤发生的分子机制

Prakasam, Gopinath; Mishra, Akhilesh; Christie, Alana; Miyata, Jeffrey; Carrillo, Deyssy; Tcheuyap, Vanina T; Ye, Hui; Do, Quyen N; Wang, Yunguan; Reig Torras, Oscar; Butti, Ramesh; Zhong, Hua; Gagan, Jeffrey; Jones, Kevin B; Carroll, Thomas J; Modrusan, Zora; Durinck, Steffen; Requena-Komuro, Mai-Carmen; Williams, Noelle S; Pedrosa, Ivan; Wang, Tao; Rakheja, Dinesh; Kapur, Payal; Brugarolas, James

A dual role for PSIP1/LEDGF in T cell acute lymphoblastic leukemia

PSIP1/LEDGF在T细胞急性淋巴细胞白血病中的双重作用

Lisa Demoen ,Filip Matthijssens ,Lindy Reunes ,Bruno Palhais ,Béatrice Lintermans ,Sara T'Sas ,Igor Fijalkowski ,Joachim Taminau ,Muluembet Z Akele ,Siska Van Belle ,Tom Taghon ,Dieter Deforce ,Filip Van Nieuwerburgh ,Geert Berx ,Panagiotis Ntziachristos ,Zeger Debyser ,Kaat Durinck ,Tim Pieters ,Steven Goossens ,Pieter Van Vlierberghe

Molecular underpinnings of dedifferentiation and aggressiveness in chromophobe renal cell carcinoma

嫌色性肾细胞癌去分化和侵袭性的分子基础

Payal Kapur, Hua Zhong, Daniel Le, Ratna Mukhopadhyay, Jeffrey Miyata, Deyssy Carrillo, Dinesh Rakheja, Satwik Rajaram, Steffen Durinck, Zora Modrusan, James Brugarolas

Assessing a single-cell multi-omic analytic platform to characterize ex vivo-engineered T-cell therapy products

评估单细胞多组学分析平台在体外工程化T细胞治疗产品表征中的应用

Maryam Moshref ,Jerry Hung-Hao Lo ,Andrew McKay ,Julien Camperi ,Joseph Schroer ,Norikiyo Ueno ,Shu Wang ,Saurabh Gulati ,Somayeh Tarighat ,Steffen Durinck ,Ho Young Lee ,Dayue Chen