日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

TR-FRET between engineered nanobodies reveals the existence of endogenous CXCR4 oligomers

利用工程纳米抗体之间的时间分辨荧光共振能量转移(TR-FRET)技术揭示了内源性CXCR4寡聚体的存在。

Heuninck, Joyce; Bobkov, Vladimir; Grison, Claire M; Fumagalli, Amos; Lescuyer, Mathias; Otun, Omolade; Bechara, Cherine; Lamarque, Laurent; Trinquet, Eric; Bachelerie, Françoise; Marin, Philippe; Mouillac, Bernard; Granier, Sébastien; van der Woning, Bas; de Haard, Hans; Smit, Martine J; Heukers, Raimond; Durroux, Thierry

A near-infrared fluorogenic dimer enables background-free imaging of endogenous GPCRs in living mice

一种近红外荧光二聚体能够对活体小鼠体内的内源性GPCR进行无背景成像

Esteoulle, Lucie; Daubeuf, François; Collot, Mayeul; Riché, Stéphanie; Durroux, Thierry; Brasse, David; Marchand, Patrice; Karpenko, Iuliia A; Klymchenko, Andrey S; Bonnet, Dominique

Pharmacological evidence for a metabotropic glutamate receptor heterodimer in neuronal cells.

神经元细胞中代谢型谷氨酸受体异二聚体的药理学证据

Moreno Delgado David, Møller Thor C, Ster Jeanne, Giraldo Jesús, Maurel Damien, Rovira Xavier, Scholler Pauline, Zwier Jurriaan M, Perroy Julie, Durroux Thierry, Trinquet Eric, Prezeau Laurent, Rondard Philippe, Pin Jean-Philippe

Structural insights into biased G protein-coupled receptor signaling revealed by fluorescence spectroscopy

荧光光谱揭示偏向性G蛋白偶联受体信号传导的结构信息

Rahmeh, Rita; Damian, Marjorie; Cottet, Martin; Orcel, Hélène; Mendre, Christiane; Durroux, Thierry; Sharma, K Shivaji; Durand, Grégory; Pucci, Bernard; Trinquet, Eric; Zwier, Jurriaan M; Deupi, Xavier; Bron, Patrick; Banères, Jean-Louis; Mouillac, Bernard; Granier, Sébastien

BRET and Time-resolved FRET strategy to study GPCR oligomerization: from cell lines toward native tissues

利用BRET和时间分辨FRET策略研究GPCR寡聚化:从细胞系到天然组织

Cottet, Martin; Faklaris, Orestis; Maurel, Damien; Scholler, Pauline; Doumazane, Etienne; Trinquet, Eric; Pin, Jean-Philippe; Durroux, Thierry

Original Fluorescent Ligand-Based Assays Open New Perspectives in G-Protein Coupled Receptor Drug Screening

原创的基于荧光配体的检测方法为G蛋白偶联受体药物筛选开辟了新的前景

Ollivier, Julien F; Shahrezaei, Vahid; Swain, Peter S; Cottet, Martin; Faklaris, Orestis; Zwier, Jurriaan M; Trinquet, Eric; Pin, Jean-Philippe; Durroux, Thierry

Time-resolved FRET between GPCR ligands reveals oligomers in native tissues

利用GPCR配体之间的时间分辨FRET技术揭示天然组织中的寡聚体

Albizu, Laura; Cottet, Martin; Kralikova, Michaela; Stoev, Stoytcho; Seyer, René; Brabet, Isabelle; Roux, Thomas; Bazin, Hervé; Bourrier, Emmanuel; Lamarque, Laurent; Breton, Christophe; Rives, Marie-Laure; Newman, Amy; Javitch, Jonathan; Trinquet, Eric; Manning, Maurice; Pin, Jean-Philippe; Mouillac, Bernard; Durroux, Thierry

Leukotriene BLT2 receptor monomers activate the G(i2) GTP-binding protein more efficiently than dimers

白三烯BLT2受体单体比二聚体更有效地激活G(i2) GTP结合蛋白。

Arcemisbéhère, Laure; Sen, Tuhinadri; Boudier, Laure; Balestre, Marie-Noëlle; Gaibelet, Gérald; Detouillon, Emilie; Orcel, Hélène; Mendre, Christiane; Rahmeh, Rita; Granier, Sébastien; Vivès, Corinne; Fieschi, Franck; Damian, Marjorie; Durroux, Thierry; Banères, Jean-Louis; Mouillac, Bernard

Building a new conceptual framework for receptor heteromers

构建受体异聚体的新概念框架

Ferré, Sergi; Baler, Ruben; Bouvier, Michel; Caron, Marc G; Devi, Lakshmi A; Durroux, Thierry; Fuxe, Kjell; George, Susan R; Javitch, Jonathan A; Lohse, Martin J; Mackie, Ken; Milligan, Graeme; Pfleger, Kevin D G; Pin, Jean-Philippe; Volkow, Nora D; Waldhoer, Maria; Woods, Amina S; Franco, Rafael

Biased agonist pharmacochaperones of the AVP V2 receptor may treat congenital nephrogenic diabetes insipidus

AVP V2受体的偏向性激动剂药理伴侣可能用于治疗先天性肾性尿崩症

Jean-Alphonse, Frédéric; Perkovska, Sanja; Frantz, Marie-Céline; Durroux, Thierry; Méjean, Catherine; Morin, Denis; Loison, Stéphanie; Bonnet, Dominique; Hibert, Marcel; Mouillac, Bernard; Mendre, Christiane