日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

XMT-2056, a HER2-Directed STING Agonist Antibody-Drug Conjugate, Induces Innate Antitumor Immune Responses by Acting on Cancer Cells and Tumor-Resident Immune Cells.

XMT-2056 是一种 HER2 靶向 STING 激动剂抗体药物偶联物,通过作用于癌细胞和肿瘤驻留免疫细胞来诱导先天性抗肿瘤免疫反应

Bukhalid Raghida A, Duvall Jeremy R, Lancaster Kelly, Catcott Kalli C, Malli Cetinbas Naniye, Monnell Travis, Routhier Caitlin, Thomas Joshua D, Bentley Keith W, Collins Scott D, Ditty Elizabeth, Eitas Timothy K, Kelleher Eugene W, Shaw Pamela, Soomer-James Jahna, Ter-Ovanesyan Elena, Xu Ling, Zurita Jeffrey, Toader Dorin, Damelin Marc, Lowinger Timothy B

Diversity-oriented synthesis yields novel multistage antimalarial inhibitors.

多样性导向合成产生新型多阶段抗疟疾抑制剂

Kato Nobutaka, Comer Eamon, Sakata-Kato Tomoyo, Sharma Arvind, Sharma Manmohan, Maetani Micah, Bastien Jessica, Brancucci Nicolas M, Bittker Joshua A, Corey Victoria, Clarke David, Derbyshire Emily R, Dornan Gillian L, Duffy Sandra, Eckley Sean, Itoe Maurice A, Koolen Karin M J, Lewis Timothy A, Lui Ping S, Lukens Amanda K, Lund Emily, March Sandra, Meibalan Elamaran, Meier Bennett C, McPhail Jacob A, Mitasev Branko, Moss Eli L, Sayes Morgane, Van Gessel Yvonne, Wawer Mathias J, Yoshinaga Takashi, Zeeman Anne-Marie, Avery Vicky M, Bhatia Sangeeta N, Burke John E, Catteruccia Flaminia, Clardy Jon C, Clemons Paul A, Dechering Koen J, Duvall Jeremy R, Foley Michael A, Gusovsky Fabian, Kocken Clemens H M, Marti Matthias, Morningstar Marshall L, Munoz Benito, Neafsey Daniel E, Sharma Amit, Winzeler Elizabeth A, Wirth Dyann F, Scherer Christina A, Schreiber Stuart L

Diversity-oriented synthesis-facilitated medicinal chemistry: toward the development of novel antimalarial agents

以多样性为导向的合成促进药物化学:迈向新型抗疟药物的开发

Comer, Eamon; Beaudoin, Jennifer A; Kato, Nobutaka; Fitzgerald, Mark E; Heidebrecht, Richard W; Lee, Maurice duPont 4th; Masi, Daniela; Mercier, Marion; Mulrooney, Carol; Muncipinto, Giovanni; Rowley, Ann; Crespo-Llado, Keila; Serrano, Adelfa E; Lukens, Amanda K; Wiegand, Roger C; Wirth, Dyann F; Palmer, Michelle A; Foley, Michael A; Munoz, Benito; Scherer, Christina A; Duvall, Jeremy R; Schreiber, Stuart L

Diversity-oriented synthesis yields a new drug lead for treatment of chagas disease

多样性导向合成法获得了一种治疗恰加斯病的新药先导化合物

Dandapani, Sivaraman; Germain, Andrew R; Jewett, Ivan; le Quement, Sebastian; Marie, Jean-Charles; Muncipinto, Giovanni; Duvall, Jeremy R; Carmody, Leigh C; Perez, Jose R; Engel, Juan C; Gut, Jiri; Kellar, Danielle; Siqueira-Neto, Jair Lage; McKerrow, James H; Kaiser, Marcel; Rodriguez, Ana; Palmer, Michelle A; Foley, Michael; Schreiber, Stuart L; Munoz, Benito

Synthesis and profiling of a diverse collection of azetidine-based scaffolds for the development of CNS-focused lead-like libraries

合成和分析多种基于氮杂环丁烷的骨架化合物,用于开发针对中枢神经系统的先导化合物库

Lowe, Jason T; Lee, Maurice D 4th; Akella, Lakshmi B; Davoine, Emeline; Donckele, Etienne J; Durak, Landon; Duvall, Jeremy R; Gerard, Baudouin; Holson, Edward B; Joliton, Adrien; Kesavan, Sarathy; Lemercier, Berenice C; Liu, Haibo; Marié, Jean-Charles; Mulrooney, Carol A; Muncipinto, Giovanni; Welzel-O'Shea, Morgan; Panko, Laura M; Rowley, Ann; Suh, Byung-Chul; Thomas, Meryl; Wagner, Florence F; Wei, Jingqiang; Foley, Michael A; Marcaurelle, Lisa A

Practical asymmetric synthesis of β-hydroxy γ-amino acids via complimentary aldol reactions

利用互补的羟醛反应实现β-羟基γ-氨基酸的实用不对称合成

Pandya, Bhaumik A; Dandapani, Sivaraman; Duvall, Jeremy R; Rowley, Ann; Mulrooney, Carol A; Ryba, Troy; Dombrowski, Michael; Harton, Marie; Young, Damian W; Marcaurelle, Lisa A