日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Covalent Protein Inhibitors via Tyrosine and Tryptophan Conjugation with Cyclic Imine Mannich Electrophiles

通过酪氨酸和色氨酸与环状亚胺曼尼希亲电试剂的共价结合制备共价蛋白抑制剂

Wang, Sijie; Wang, Lei; Hadisurya, Marco; Nia, Siavash Shahbazi; Tao, W Andy; Dykhuizen, Emily C; Krusemark, Casey J

Structural landscape of H3K27me3 recognition by protein domains and their potential for inhibition

蛋白质结构域识别H3K27me3的结构图谱及其抑制潜力

Rosas, Ruben; Baracaldo-Lancheros, Luisa F; Dykhuizen, Emily C; Musselman, Catherine A

PBRM1-Dependent PBAF Targeting is Required for EMT and Metastasis in Breast Cancer

PBRM1依赖性PBAF靶向是乳腺癌EMT和转移所必需的

Dhiman, Alisha; Ayers, Mitchell G; McCuiston, Jamie L; Shinde, Aparna B; Akhand, Saeed Salehin; Jiao, Guanming; Jauregui-Lozano, Juan; Hadisurya, Marco; Porter, Elizabeth G; Tao, W Andy; Weake, Vikki M; Zhang, Yucheng; Utturkar, Sagar M; Maraunde, Matthew R; Wendt, Michael K; Dykhuizen, Emily C

KRAS-mediated upregulation of CIP2A promotes suppression of PP2A-B56α to initiate pancreatic cancer development.

KRAS介导的CIP2A上调促进PP2A-B56α的抑制,从而启动胰腺癌的发展。

Tinsley Samantha L, Chianis Ella Rose D, Shelley Rebecca A, Mall Gaganpreet K, Dhiman Alisha, Baral Garima, Kothandaraman Harish, Thoma Mary C, English Isabel A, Daniel Colin J, Acosta Luis Carlos Sanjuan, Solorio Luis, Atallah Lanman Nadia, Pasca di Magliano Marina, Narla Goutham, Dykhuizen Emily C, Sears Rosalie C, Allen-Petersen Brittany L

Activity-assembled nBAF complex mediates rapid immediate early gene transcription by regulating RNA polymerase II productive elongation.

活性组装的 nBAF 复合物通过调节 RNA 聚合酶 II 的有效延伸来介导快速的早期基因转录

Cornejo Karen G, Venegas Andie, Sono Morgan H, Door Madeline, Gutierrez-Ruiz Brenda, Karabedian Lucy B, Nandi Supratik G, Hadisurya Marco, Tao W Andy, Dykhuizen Emily C, Saha Ramendra N

MicroRNA-directed pathway discovery elucidates an miR-221/222-mediated regulatory circuit in class switch recombination

微RNA指导的通路发现阐明了miR-221/222介导的类别转换重组调控回路

Wigton, Eric J; Mikami, Yohei; McMonigle, Ryan J; Castellanos, Carlos A; Wade-Vallance, Adam K; Zhou, Simon K; Kageyama, Robin; Litterman, Adam; Roy, Suparna; Kitamura, Daisuke; Dykhuizen, Emily C; Allen, Christopher D C; Hu, Hui; O'Shea, John J; Ansel, K Mark

At the Crossroad of Gene Regulation and Genome Organization: Potential Roles for ATP-Dependent Chromatin Remodelers in the Regulation of CTCF-Mediated 3D Architecture

基因调控与基因组组织交汇点:ATP依赖性染色质重塑因子在CTCF介导的三维结构调控中的潜在作用

Alpsoy, Aktan; Sood, Surbhi; Dykhuizen, Emily C

Polycomb Paralog Chromodomain Inhibitors Active against Both CBX6 and CBX8*

对CBX6和CBX8均有活性的多梳蛋白旁系同源染色质结构域抑制剂*

Milosevich, Natalia; Wilson, Chelsea R; Brown, Tyler M; Alpsoy, Aktan; Wang, Sijie; Connelly, Katelyn E; Sinclair, Kirsten A D; Ponio, Felino R; Hof, Rebecca; Dykhuizen, Emily C; Hof, Fraser

Polycomb group proteins in cancer: multifaceted functions and strategies for modulation

多梳蛋白在癌症中的作用:多重功能及调控策略

Wang, Sijie; C Ordonez-Rubiano, Sandra; Dhiman, Alisha; Jiao, Guanming; Strohmier, Brayden P; Krusemark, Casey J; Dykhuizen, Emily C

A Potent, Selective CBX2 Chromodomain Ligand and Its Cellular Activity During Prostate Cancer Neuroendocrine Differentiation

一种强效、选择性的CBX2染色质结构域配体及其在前列腺癌神经内分泌分化过程中的细胞活性

Wang, Sijie; Alpsoy, Aktan; Sood, Surbhi; Ordonez-Rubiano, Sandra Carolina; Dhiman, Alisha; Sun, Yixing; Jiao, Guanming; Krusemark, Casey J; Dykhuizen, Emily C