Bile acids target an exposed cavity in the glucocorticoid receptor modulating receptor self-assembly, chromatin binding and transcriptional activity
胆汁酸靶向糖皮质激素受体上暴露的空腔,从而调节受体的自组装、染色质结合和转录活性。
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doi:10.1101/2025.05.13.653693
Jiménez-Panizo, Alba; Johnson, Thomas A; Wagh, Kaustubh; Alegre-Martí, Andrea; Novoa, Inés Montoya; Lafuente, Agustina L; Eckhard, Ulrich; Rodríguez-Lumbreras, Luis Ángel; Hoang, Le; Stortz, Martín; Abella, Montserrat; Goldstein, Ido; Valledor-Fernández, Annabel; Varticovski, Lyuba; Arias, Irwin; Presman, Diego M; Stavreva, Diana A; Fernández-Recio, Juan; Fuentes-Prior, Pablo; Hager, Gordon L; Estébanez-Perpiñá, Eva