日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

FlowMol3: flow matching for 3D de novo small-molecule generation

FlowMol3:用于三维从头小分子生成的流动匹配

Moumad, Aziz; Bouhaoui, Abderrazzak; Eddahmi, Mohammed; Catto, Marco; Bouissane, Latifa; Dunn, Ian; Koes, David R

Experimental and MEDT Study of Sydnone–Alkyne Cycloaddition-Based Synthesis of 1,4-Disubstituted Pyrazoles and In Silico Investigation of Their Binding to HCV and HIV Proteins

基于炔酮-炔环加成反应合成1,4-二取代吡唑的实验和MEDT研究及其与HCV和HIV蛋白结合的计算机模拟研究

Lee, Jin; Park, Jongha; Park, Jino; Park, Yong Eun; Choi, Joon Hyuk; Heo, Nae-Yun; Park, Seung Ha; Kim, Tae Oh; Zerbib, Souad; Eddahmi, Mohammed; Alaqarbeh, Marwa; Bodet, Pierre-Edouard; Thiery, Valérie; Fatimi, Ahmed; Cruz-Martins, Natália; Bailly, Christian; Domingo, Luis R; Bouissane, Latifa

Synthesis, Molecular Electron Density Theory Study, Molecular Docking, and Pharmacological Evaluation of New Coumarin-Sulfonamide-Nitroindazolyl-Triazole Hybrids as Monoamine Oxidase Inhibitors.

新型香豆素-磺酰胺-硝基吲唑基-三唑杂合物作为单胺氧化酶抑制剂的合成、分子电子密度理论研究、分子对接和药理学评价

Eddahmi Mohammed, La Spada Gabriella, Domingo Luis R, Vergoten Gérard, Bailly Christian, Catto Marco, Bouissane Latifa

A Suitable Functionalization of Nitroindazoles with Triazolyl and Pyrazolyl Moieties via Cycloaddition Reactions

通过环加成反应对硝基吲唑进行合适的三唑基和吡唑基官能化

Eddahmi, Mohammed; Moura, Nuno M M; Bouissane, Latifa; Amiri, Ouafa; Faustino, M Amparo F; Cavaleiro, José A S; Mendes, Ricardo F; Paz, Filipe A A; Neves, Maria G P M S; Rakib, El Mostapha