日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

2-Aminothiophene Derivative SB-83 Inhibits Trypanothione Reductase and Modulates Cytokine Production in Trypanosoma cruzi-Infected Cells

2-氨基噻吩衍生物SB-83抑制锥虫硫还原酶并调节克氏锥虫感染细胞中的细胞因子产生

Dos Santos, Airton Lucas Sousa; de Souza, Vanessa Maria Rodrigues; de Sousa, Julyanne Maria Saraiva; Rodrigues, Raiza Raianne Luz; Braga, Mércya Lopes; Da Silva Sousa, Maria Gabrielly Gonçalves; de Oliveira, Douglas Soares; da Silva, Mirely Vitória Farias; da Silva-Junior, Edeildo Ferreira; de Lima Nunes, Thaís Amanda; da Silva, Marcos Vinícius; da Silva, Ingrid Gracielle Martins; Barros-Cordeiro, Karine Brenda; Báo, Sônia Nair; Mendonça Junior, Francisco Jaime Bezerra; da Franca Rodrigues, Klinger Antonio

Modifying Antibiotic Activity of Synthetic Thiadiazine Analogs Against MDR Bacteria and ADMET Analysis

合成噻二嗪类似物对多重耐药菌的抗菌活性修饰及ADMET分析

de Oliveira Borges, João Arthur; Freitas, Priscilla Ramos; Araújo, Isaac Moura; de Almeida, Ray Silva; Dos Santos Nascimento, Igor José; de Araújo-Júnior, João Xavier; da Silva-Júnior, Edeildo Ferreira; de Aquino, Thiago Mendonça; Junior, Francisco Jaime Bezerra Mendonça; Marinho, Emmanuel Silva; Dos Santos, Hélcio Silva; Kowalski, Radosław; Kowalska, Grażyna; Coutinho, Henrique Douglas Melo; Tintino, Saulo Relison; de Araújo, Ana Carolina Justino

Bifenthrin Under Scrutiny: Revisiting Toxicological Evidence Amid Regulatory Gaps

联苯菊酯面临审查:监管漏洞下的毒理学证据再探

Moreira, Caroline V L; Ogbu, John 1st; Monteiro, Kadja L C; de Aquino, Thiago M; da Silva-Júnior, Edeildo F; Filho, Alberto S S; Napolitano, Hamilton B; Elusiyan, Christianah A; do Couto, Renê O; Costa, Elson A; Fajemiroye, James O

Evaluation of the Efflux Pump Inhibition Activity of Thiadiazine-Derived Compounds Against the Staphylococcus aureus 1199B Strain

评价噻二嗪类化合物对金黄色葡萄球菌1199B菌株的外排泵抑制活性

Roque Paulo, Cicera Laura; Alexandre, Priscilla Ramos Freitas; Araujo, Ana Carolina Ferreira; Almeida, Ray Silva; Albuquerque, Emílio Sousa; Oliveira-Tintino, Cícera Datiane de Morais; Nascimento, Igor J S; Araújo-Júnior, João Xavier; Silva-Junior, Edeildo Ferreira da; Aquino, Thiago Mendonça de; Mendonça-Junior, Francisco Jaime Bezerra; Araújo-Neto, José Bezerra de; Silva Leandro, Maria Karollyna do Nascimento; Menezes, Irwin Rose Alencar de; Coutinho, Henrique Douglas Melo; Rocha, Janaina Esmeraldo

New Cinnamamide and Derivatives as New Larvicides against Aedes aegypti Vector Larvae: Facile Synthesis, In Silico Study, In Vitro Noncytotoxicity, and Nontoxicity against Zebrafish

新型肉桂酰胺及其衍生物作为新型杀幼虫剂对抗埃及伊蚊幼虫:简易合成、计算机模拟研究、体外无细胞毒性及对斑马鱼无毒性

da Silva, Adrielle Firmino; França, Saraliny Bezerra; Ferreira, Erick Gabriel Alves; de Oliveira Barreto, Emiliano; Mclaine Duarte de Freitas, Jeniffer; Duarte de Freitas, Johnnatan; da Silva Júnior, Edeildo Ferreira; Leite, Ana Catarina Rezende; Dos Santos, Pedro Correia Gomes; de Azevedo, Rafael David Souto; da Silva, Josefa Gerlane; da Paz Lima, Dimas José

Antidiabetic Activity and Inhibitory Effects of Derivatives of Advanced Aminoguanidine Glycation

高级氨基胍糖苷衍生物的抗糖尿病活性和抑制作用

Sarmento, Patrícia de Albuquerque; da Silva, Andressa Letícia Lopes; Ferreira da Silva-Júnior, Edeildo; Scio, Elita; Aragão, Danielle Maria de Oliveira; Ribeiro, Êurica Adélia Nogueira; Rodrigues, Érica Erlanny da Silva; Aquino, Pedro Gregório Vieira; Santos, Bárbara Viviana de Oliveira; Santana, Antônio Euzébio Goulart; de Queiroz, Aline Cavalcanti; Alexandre-Moreira, Magna Suzana; Coutinho, Henrique Douglas Melo; de Araújo Júnior, João Xavier

Insights on Natural Products Against Amyotrophic Lateral Sclerosis (ALS)

天然产物对抗肌萎缩侧索硬化症(ALS)的研究进展

Monteiro, Kadja Luana Chagas; Dos Santos Alcântara, Marcone Gomes; de Aquino, Thiago Mendonça; da Silva-Júnior, Edeildo Ferreira

Emerging drug design strategies in anti-influenza drug discovery

抗流感药物研发中新兴的药物设计策略

Liu, Chuanfeng; Hu, Lide; Dong, Guanyu; Zhang, Ying; Ferreira da Silva-Júnior, Edeildo; Liu, Xinyong; Menéndez-Arias, Luis; Zhan, Peng

Development of chalcone-like derivatives and their biological and mechanistic investigations as novel influenza nuclear export inhibitors

查尔酮类衍生物的开发及其作为新型流感核输出抑制剂的生物学和机制研究

Chuanfeng Liu, Ying Zhang, Ping Li, Huinan Jia, Han Ju, Jiwei Zhang, Edeildo Ferreira da Silva-Júnior, Sunanda Samanta, Parimal Kar, Bing Huang, Xinyong Liu, Peng Zhan

Coumarin-Based Compounds as Inhibitors of Tyrosinase/Tyrosine Hydroxylase: Synthesis, Kinetic Studies, and In Silico Approaches

香豆素类化合物作为酪氨酸酶/酪氨酸羟化酶抑制剂:合成、动力学研究和计算机模拟方法

Jéssica Alves Nunes, Rodrigo Santos Aquino de Araújo, Fabrícia Nunes da Silva, Joanna Cytarska, Krzysztof Z Łączkowski, Sílvia Helena Cardoso, Francisco Jaime Bezerra Mendonça-Júnior, Edeildo Ferreira da Silva-Júnior