Bexarotene Binds to the Amyloid Precursor Protein Transmembrane Domain, Alters Its α-Helical Conformation, and Inhibits γ-Secretase Nonselectively in Liposomes
贝沙罗汀与淀粉样蛋白前体跨膜结构域结合,改变其 α-螺旋构象,并在脂质体中非选择性地抑制 γ-分泌酶
期刊:ACS Chemical Neuroscience
影响因子:4.1
doi:10.1021/acschemneuro.8b00068
Frits Kamp, Holger A Scheidt, Edith Winkler, Gabriele Basset, Hannes Heinel, James M Hutchison, Loren M LaPointe, Charles R Sanders, Harald Steiner, Daniel Huster