日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

High-affinity, structure-validated and selective macrocyclic peptide tools for chemical biology studies of Huntingtin

用于亨廷顿蛋白化学生物学研究的高亲和力、结构验证和选择性大环肽工具

Fanti, Rebeka; Wolf, Esther; Ikenoue, Tatsuya; Deme, Justin C; Balakrishnan, Swati; Keith, Brandon A; Alteen, Matthew G; Chandrasekaran, Renu; Yadav, Manisha; Bhajiawala, Ritika; Ackloo, Suzanne; Feng, Jia; Pouladi, Mahmoud A; Edwards, Aled M; Wilson, Derek J; Lea, Susan M; Suga, Hiroaki; Harding, Rachel J

CACHE Challenge #3: Targeting the Nsp3 Macrodomain of SARS-CoV-2

CACHE挑战赛#3:靶向SARS-CoV-2的Nsp3宏结构域

Herasymenko, Oleksandra; Silva, Madhushika; Correy, Galen J; Abu-Saleh, Abd Al-Aziz A; Ackloo, Suzanne; Arrowsmith, Cheryl; Ashworth, Alan; Ban, Fuqiang; Beck, Hartmut; Bishop, Kevin P; Bohórquez, Hugo J; Bolotokova, Albina; Breznik, Marko; Chau, Irene; Chen, Yu; Cherkasov, Artem; Dehaen, Wim; Della Corte, Dennis; Denzinger, Katrin; Doering, Niklas P; Edfeldt, Kristina; Edwards, Aled; Fayne, Darren; Gentile, Francesco; Gibson, Elisa; Gokdemir, Ozan; Gunnarsson, Anders; Günther, Judith; Irwin, John J; Jensen, Jan Halborg; Harding, Rachel J; Hillisch, Alexander; Hoffer, Laurent; Hogner, Anders; Hutchinson, Ashley; Kandwal, Shubhangi; Karlova, Andrea; Koirala, Kushal; Kotelnikov, Sergei; Kozakov, Dima; Lee, Juyong; Lee, Soowon; Lessel, Uta; Liu, Sijie; Liu, Xuefeng; Loppnau, Peter; Meiler, Jens; Moretti, Rocco; Moroz, Yurii S; Muvva, Charuvaka; Oprea, Tudor I; Paige, Brooks; Pandit, Amit; Park, Keunwan; Poda, Gennady; Protopopov, Mykola V; Pütter, Vera; Ravichandran, Rahul; Rognan, Didier; Rosta, Edina; Sabnis, Yogesh; Scott, Thomas; Seitova, Almagul; Sharma, Purshotam; Sindt, François; Song, Minghu; Steinmann, Casper; Stevens, Rick; Talagayev, Valerij; Tararina, Valentyna V; Tarkhanova, Olga; Tingey, Damon; Trant, John F; Treleaven, Dakota; Tropsha, Alexander; Walters, Patrick; Wells, Jude; Westermaier, Yvonne; Wolber, Gerhard; Wortmann, Lars; Zheng, Shuangjia; Fraser, James S; Schapira, Matthieu

A consensus platform for antibody characterization.

抗体表征的共识平台。

Ayoubi Riham, Ryan Joel, Gonzalez Bolivar Sara, Alende Charles, Ruiz Moleon Vera, Fotouhi Maryam, Alqazzaz Mona, Southern Kathleen, Alshafie Walaa, Baker Matt R, Ball Alexander R Jr, Callahan Danielle, Cooper Jeffery A, Crosby Katherine, Harvey Kevin J, Houston Douglas W, Kumaran Ravindran, Rego Meghan, Schofield Christine, Wu Hai, Biddle Michael S, Brown Claire M, Kahn Richard A, Bandrowski Anita, Virk Harvinder S, Edwards Aled M, McPherson Peter S, Laflamme Carl

Enantioselective protein affinity selection mass spectrometry (E-ASMS)

对映选择性蛋白质亲和力选择质谱法(E-ASMS)

Wang, Xiaoyun; Sun, Jianxian; Ahmad, Shabbir; Yang, Diwen; Li, Fengling; Chan, U Hang; Zeng, Hong; Simoben, Conrad V; Green, Stuart R; Silva, Madhushika; Houliston, Scott; Dong, Aiping; Bolotokova, Albina; Gibson, Elisa; Kutera, Maria; Ghiabi, Pegah; Kondratov, Ivan; Matviyuk, Tetiana; Chuprina, Alexander; Mavridi, Danai; Lenz, Christopher; Joerger, Andreas C; Brown, Benjamin D; Heath, Richard B; Yue, Wyatt W; Robbie, Lucy K; Beyett, Tyler S; Müller, Susanne; Knapp, Stefan; Owen, Dafydd R; Harding, Rachel; Schapira, Matthieu; Brown, Peter J; Santhakumar, Vijayaratnam; Ackloo, Suzanne; Arrowsmith, Cheryl H; Edwards, Aled M; Peng, Hui; Halabelian, Levon

Structural basis of TMPRSS11D specificity and autocleavage activation.

TMPRSS11D 特异性和自切割激活的结构基础

Fraser Bryan J, Wilson Ryan P, Ferková Sára, Ilyassov Olzhas, Lac Jackie, Dong Aiping, Li Yen-Yen, Seitova Alma, Li Yanjun, Hejazi Zahra, Kenney Tristan M G, Penn Linda Z, Edwards Aled, Leduc Richard, Boudreault Pierre-Luc, Morin Gregg B, Bénard François, Arrowsmith Cheryl H

The Chemical Probes Portal - 2024: update on this public resource to support best-practice selection and use of small molecules in biomedical research

化学探针门户网站 - 2024:更新此公共资源,以支持生物医学研究中小分子的最佳实践选择和使用

Sanfelice, Domenico; Antolin, Albert A; Crisp, Alisa; Chen, Yi; Bellenie, Benjamin; Brennan, Paul E; Edwards, Aled; Müller, Susanne; Al-Lazikani, Bissan; Workman, Paul

A Target Class Ligandability Evaluation of WD40 Repeat-Containing Proteins

WD40重复序列蛋白的靶向配体结合能力评价

Ackloo, Suzanne; Li, Fengling; Szewczyk, Magda; Seitova, Almagul; Loppnau, Peter; Zeng, Hong; Xu, Jin; Ahmad, Shabbir; Arnautova, Yelena A; Baghaie, A J; Beldar, Serap; Bolotokova, Albina; Centrella, Paolo A; Chau, Irene; Clark, Matthew A; Cuozzo, John W; Dehghani-Tafti, Saba; Disch, Jeremy S; Dong, Aiping; Dumas, Antoine; Feng, Jianwen A; Ghiabi, Pegah; Gibson, Elisa; Gilmer, Justin; Goldman, Brian; Green, Stuart R; Guié, Marie-Aude; Guilinger, John P; Harms, Nathan; Herasymenko, Oleksandra; Houliston, Scott; Hutchinson, Ashley; Kearnes, Steven; Keefe, Anthony D; Kimani, Serah W; Kramer, Trevor; Kutera, Maria; Kwak, Haejin A; Lento, Cristina; Li, Yanjun; Liu, Jenny; Loup, Joachim; Machado, Raquel A C; Mulhern, Christopher J; Perveen, Sumera; Righetto, Germanna L; Riley, Patrick; Shrestha, Suman; Sigel, Eric A; Silva, Madhushika; Sintchak, Michael D; Slakman, Belinda L; Taylor, Rhys D; Thompson, James; Torng, Wen; Underkoffler, Carl; von Rechenberg, Moritz; Walsh, Ryan T; Watson, Ian; Wilson, Derek J; Wolf, Esther; Yadav, Manisha; Yazdi, Aliakbar K; Zhang, Junyi; Zhang, Ying; Santhakumar, Vijayaratnam; Edwards, Aled M; Barsyte-Lovejoy, Dalia; Schapira, Matthieu; Brown, Peter J; Halabelian, Levon; Arrowsmith, Cheryl H

Enabling Open Machine Learning of Deoxyribonucleic Acid-Encoded Library Selections to Accelerate the Discovery of Small Molecule Protein Binders

利用开放式机器学习对脱氧核糖核酸编码文库进行筛选,加速小分子蛋白质结合剂的发现

Wellnitz, James; Ahmad, Shabbir; Bagale, Nabin; Cheng, Xuemin; Joseph, Jermiah; Zeng, Hong; Bolotokova, Albina; Dong, Aiping; Reza, Shaghayegh; Ghiabi, Pegah; Gibson, Elisa; Tu, Guiping; Li, Xianyang; Liu, Jian; Dou, Dengfeng; Li, Jin; Foley, Timothy L; Harris, Anthony R; Klug-McLeod, Jacquelyn L; Lee, Jisun; Lengyel-Zhand, Zsofia; Montgomery, Justin I; Sakata, Sylvie; Zhang, Jinzhi; Zhu, Hongyao; Owen, Dafydd R; Harding, Rachel J; Edwards, Aled M; Haibe-Kains, Benjamin; Halabelian, Levon; Tropsha, Alexander; Couñago, Rafael M

CACHE Challenge #2: Targeting the RNA Site of the SARS-CoV-2 Helicase Nsp13

CACHE挑战#2:靶向SARS-CoV-2解旋酶Nsp13的RNA位点

Herasymenko, Oleksandra; Silva, Madhushika; Abu-Saleh, Abd Al-Aziz A; Ahmad, Ayaz; Alvarado-Huayhuaz, Jesus; Arce, Oscar E A; Armstrong, Roly J; Arrowsmith, Cheryl; Bachta, Kelly E; Beck, Hartmut; Berta, Denes; Bieniek, Mateusz K; Blay, Vincent; Bolotokova, Albina; Bourne, Philip E; Breznik, Marko; Brown, Peter J; Campbell, Aaron D G; Carosati, Emanuele; Chau, Irene; Cole, Daniel J; Cree, Ben; Dehaen, Wim; Denzinger, Katrin; Dos Santos Machado, Karina; Dunn, Ian; Durai, Prasannavenkatesh; Edfeldt, Kristina; Edwards, Aled; Fayne, Darren; Felfoldi, Daniel; Friston, Kallie; Ghiabi, Pegah; Gibson, Elisa; Günther, Judith; Gunnarsson, Anders; Hillisch, Alexander; Houston, Douglas R; Jensen, Jan Halborg; Harding, Rachel J; Harris, Kate S; Hoffer, Laurent; Hogner, Anders; Horton, Joshua T; Houliston, Scott; Hultquist, Judd F; Hutchinson, Ashley; Irwin, John J; Jukič, Marko; Kandwal, Shubhangi; Karlova, Andrea; Katis, Vittorio L; Kich, Ryan P; Kireev, Dmitri; Koes, David; Inniss, Nicole L; Lessel, Uta; Liu, Sijie; Loppnau, Peter; Lu, Wei; Martino, Sam; McGibbon, Miles; Meiler, Jens; Mettu, Akhila; Money-Kyrle, Sam; Moretti, Rocco; Moroz, Yurii S; Muvva, Charuvaka; Newman, Joseph A; Obendorf, Leon; Paige, Brooks; Pandit, Amit; Park, Keunwan; Perveen, Sumera; Pirie, Rachael; Poda, Gennady; Protopopov, Mykola; Pütter, Vera; Ricci, Federico; Roper, Natalie J; Rosta, Edina; Rzhetskaya, Margarita; Sabnis, Yogesh; Satchell, Karla J F; Schmitt Kremer, Frederico; Scott, Thomas; Seitova, Almagul; Steinmann, Casper; Talagayev, Valerij; Tarkhanova, Olga O; Tatum, Natalie J; Treleaven, Dakota; Velasque Werhli, Adriano; Walters, W Patrick; Wang, Xiaowen; Wells, Jude; Wells, Geoffrey; Westermaier, Yvonne; Wolber, Gerhard; Wortmann, Lars; Zhang, Jixian; Zhao, Zheng; Zheng, Shuangjia; Schapira, Matthieu

Toward target 2035: EUbOPEN - a public-private partnership to enable & unlock biology in the open

迈向2035年目标:EUbOPEN——一项旨在促进和开放生物学的公私合作项目

Tredup, Claudia; Ackloo, Suzanne; Beck, Hartmut; Brown, Peter J; Bullock, Alex N; Ciulli, Alessio; Dikic, Ivan; Edfeldt, Kristina; Edwards, Aled M; Elkins, Jonathan M; Farin, Henner F; Fon, Edward A; Gstaiger, Matthias; Günther, Judith; Gustavsson, Anna-Lena; Häberle, Sandra; Isigkeit, Laura; Huber, Kilian V M; Kotschy, Andras; Krämer, Oliver; Leach, Andrew R; Marsden, Brian D; Matsui, Hisanori; Merk, Daniel; Montel, Florian; Mulder, Monique P C; Müller, Susanne; Owen, Dafydd R; Proschak, Ewgenij; Röhm, Sandra; Stolz, Alexandra; Sundström, Michael; von Delft, Frank; Willson, Timothy M; Arrowsmith, Cheryl H; Knapp, Stefan