日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization of Covalent MKK7 Inhibitors via Crude Nanomole-Scale Libraries

通过粗纳摩尔级库优化共价 MKK7 抑制剂

Paul Gehrtz, Shir Marom, Mike Bührmann, Julia Hardick, Silke Kleinbölting, Amit Shraga, Christian Dubiella, Ronen Gabizon, Jan N Wiese, Matthias P Müller, Galit Cohen, Ilana Babaev, Khriesto Shurrush, Liat Avram, Efrat Resnick, Haim Barr, Daniel Rauh, Nir London

Tunable Methacrylamides for Covalent Ligand Directed Release Chemistry

用于共价配体定向释放化学的可调甲基丙烯酰胺

Rambabu N Reddi ,Efrat Resnick ,Adi Rogel ,Boddu Venkateswara Rao ,Ronen Gabizon ,Kim Goldenberg ,Neta Gurwicz ,Daniel Zaidman ,Alexander Plotnikov ,Haim Barr ,Ziv Shulman ,Nir London

Site-Specific Labeling of Endogenous Proteins Using CoLDR Chemistry

利用CoLDR化学方法对内源性蛋白质进行位点特异性标记

Rambabu N Reddi ,Adi Rogel ,Efrat Resnick ,Ronen Gabizon ,Pragati Kishore Prasad ,Neta Gurwicz ,Haim Barr ,Ziv Shulman ,Nir London

Sulfopin is a covalent inhibitor of Pin1 that blocks Myc-driven tumors in vivo

Sulfopin 是一种 Pin1 共价抑制剂,可在体内阻断 Myc 驱动的肿瘤。

Christian Dubiella # ,Benika J Pinch # ,Kazuhiro Koikawa ,Daniel Zaidman ,Evon Poon ,Theresa D Manz ,Behnam Nabet ,Shuning He ,Efrat Resnick ,Adi Rogel ,Ellen M Langer ,Colin J Daniel ,Hyuk-Soo Seo ,Ying Chen ,Guillaume Adelmant ,Shabnam Sharifzadeh ,Scott B Ficarro ,Yann Jamin ,Barbara Martins da Costa ,Mark W Zimmerman ,Xiaolan Lian ,Shin Kibe ,Shingo Kozono ,Zainab M Doctor ,Christopher M Browne ,Annan Yang ,Liat Stoler-Barak ,Richa B Shah ,Nicholas E Vangos ,Ezekiel A Geffken ,Roni Oren ,Eriko Koide ,Samuel Sidi ,Ziv Shulman ,Chu Wang ,Jarrod A Marto ,Sirano Dhe-Paganon ,Thomas Look ,Xiao Zhen Zhou ,Kun Ping Lu ,Rosalie C Sears ,Louis Chesler ,Nathanael S Gray ,Nir London

An automatic pipeline for the design of irreversible derivatives identifies a potent SARS-CoV-2 Mpro inhibitor

不可逆衍生物设计的自动流程可识别有效的 SARS-CoV-2 Mpro 抑制剂

Daniel Zaidman, Paul Gehrtz, Mihajlo Filep, Daren Fearon, Ronen Gabizon, Alice Douangamath, Jaime Prilusky, Shirly Duberstein, Galit Cohen, C David Owen, Efrat Resnick, Claire Strain-Damerell, Petra Lukacik; Covid-Moonshot Consortium; Haim Barr, Martin A Walsh, Frank von Delft, Nir London

Rapid Covalent-Probe Discovery by Electrophile-Fragment Screening

通过亲电片段筛选快速发现共价探针

Efrat Resnick, Anthony Bradley, Jinrui Gan, Alice Douangamath, Tobias Krojer, Ritika Sethi, Paul P Geurink, Anthony Aimon, Gabriel Amitai, Dom Bellini, James Bennett, Michael Fairhead, Oleg Fedorov, Ronen Gabizon, Jin Gan, Jingxu Guo, Alexander Plotnikov, Nava Reznik, Gian Filippo Ruda, Laura Díaz-S