日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Click. Screen. Degrade. A Miniaturized D2B Workflow for Rapid PROTAC Discovery

点击。屏幕。降级。用于快速 PROTAC 发现的微型化 D2B 工作流程

Mitrović, Marko; Greco, Francesco Aleksy; García, Yiliam Cruz; Lučić, Aleksandar; Hoffmann, Lasse; Chander, Rohit; Schönfeld, Julia; Liebisch, Nick; Sivashanmugam, Saran Aswathaman; Schwalm, Martin Peter; Egner, Markus; Lewandowski, Max; Merk, Daniel; Morasch, Viktoria; Wolf, Elmar; Müller, Susanne; Hanke, Thomas; Proschak, Ewgenij; Hiesinger, Kerstin; Knapp, Stefan

De Novo Discovery of α,α-Disubstituted α-amino Acid-Containing α-helical Peptides as Competitive PPARγ PPI Inhibitors

从头发现含α,α-二取代α-氨基酸的α-螺旋肽作为竞争性PPARγ PPI抑制剂

Sigal, Maxwell; Egner, Markus; Okada, Chikako; Merk, Daniel; Sengoku, Toru; Katoh, Takayuki; Suga, Hiroaki

A Nurr1 Agonist Derived from the Natural Ligand DHI Induces Neuroprotective Gene Expression.

源自天然配体DHI的Nurr1激动剂可诱导神经保护基因表达

Egner Markus, Busch Romy, López-García Úrsula, Lewandowski Max, Höfner Georg, Wein Thomas, Marschner Julian A, Merk Daniel