日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design and Synthesis of Pyridine-Based Pyrrolo[2,3-d]pyrimidine Analogs as CSF1R Inhibitors: Molecular Hybridization and Scaffold Hopping Approach

吡啶类吡咯并[2,3-d]嘧啶类似物作为CSF1R抑制剂的设计与合成:分子杂交和骨架跃迁方法

Cherukupalli, Srinivasulu; Degenhart, Carsten; Habenberger, Peter; Unger, Anke; Eickhoff, Jan; Hoff, Bård Helge; Sundby, Eirik

Evaluating Triazole-Substituted Pyrrolopyrimidines as CSF1R Inhibitors

评价三唑取代的吡咯并嘧啶类化合物作为 CSF1R 抑制剂的活性

Cherukupalli, Srinivasulu; Eickhoff, Jan; Degenhart, Carsten; Habenberger, Peter; Unger, Anke; Hoff, Bård Helge; Sundby, Eirik

Combined Treatment with Host-Directed and Anticytomegaloviral Kinase Inhibitors: Mechanisms, Synergisms and Drug Resistance Barriers

宿主导向激酶抑制剂与抗巨细胞病毒激酶抑制剂联合治疗:机制、协同作用和耐药性障碍

Wild, Markus; Karner, Dubravka; Eickhoff, Jan; Wagner, Sabrina; Kicuntod, Jintawee; Chang, William; Barry, Peter; Jonjić, Stipan; Lenac Roviš, Tihana; Marschall, Manfred

Discovery of the Hedgehog Pathway Inhibitor Pipinib that Targets PI4KIIIß

发现靶向 PI4KIIIβ 的 Hedgehog 通路抑制剂 Pipinib

Kremer, Lea; Hennes, Elisabeth; Brause, Alexandra; Ursu, Andrei; Robke, Lucas; Matsubayashi, Hideaki T; Nihongaki, Yuta; Flegel, Jana; Mejdrová, Ivana; Eickhoff, Jan; Baumann, Matthias; Nencka, Radim; Janning, Petra; Kordes, Susanne; Schöler, Hans R; Sterneckert, Jared; Inoue, Takanari; Ziegler, Slava; Waldmann, Herbert

Dual Inhibition of GSK3β and CDK5 Protects the Cytoskeleton of Neurons from Neuroinflammatory-Mediated Degeneration In Vitro and In Vivo

双重抑制GSK3β和CDK5可在体外和体内保护神经元细胞骨架免受神经炎症介导的退行性变。

Reinhardt, Lydia; Kordes, Susanne; Reinhardt, Peter; Glatza, Michael; Baumann, Matthias; Drexler, Hannes C A; Menninger, Sascha; Zischinsky, Gunther; Eickhoff, Jan; Fröb, Claudia; Bhattarai, Prabesh; Arulmozhivarman, Guruchandar; Marrone, Lara; Janosch, Antje; Adachi, Kenjiro; Stehling, Martin; Anderson, Eric N; Abo-Rady, Masin; Bickle, Marc; Pandey, Udai Bhan; Reimer, Michell M; Kizil, Caghan; Schöler, Hans R; Nussbaumer, Peter; Klebl, Bert; Sterneckert, Jared L

Modulators of 14-3-3 Protein-Protein Interactions

14-3-3蛋白-蛋白相互作用的调节因子

Stevers, Loes M; Sijbesma, Eline; Botta, Maurizio; MacKintosh, Carol; Obsil, Tomas; Landrieu, Isabelle; Cau, Ylenia; Wilson, Andrew J; Karawajczyk, Anna; Eickhoff, Jan; Davis, Jeremy; Hann, Michael; O'Mahony, Gavin; Doveston, Richard G; Brunsveld, Luc; Ottmann, Christian

Systematic Kinase Inhibitor Profiling Identifies CDK9 as a Synthetic Lethal Target in NUT Midline Carcinoma

系统性激酶抑制剂谱分析发现 CDK9 是 NUT 中线癌的合成致死靶点

Brägelmann, Johannes; Dammert, Marcel A; Dietlein, Felix; Heuckmann, Johannes M; Choidas, Axel; Böhm, Stefanie; Richters, André; Basu, Debjit; Tischler, Verena; Lorenz, Carina; Habenberger, Peter; Fang, Zhizhou; Ortiz-Cuaran, Sandra; Leenders, Frauke; Eickhoff, Jan; Koch, Uwe; Getlik, Matthäus; Termathe, Martin; Sallouh, Muhammad; Greff, Zoltán; Varga, Zoltán; Balke-Want, Hyatt; French, Christopher A; Peifer, Martin; Reinhardt, H Christian; Örfi, László; Kéri, György; Ansén, Sascha; Heukamp, Lukas C; Büttner, Reinhard; Rauh, Daniel; Klebl, Bert M; Thomas, Roman K; Sos, Martin L

Functional classification of memory CD8(+) T cells by CX3CR1 expression

根据 CX3CR1 表达对记忆性 CD8(+) T 细胞进行功能分类

Jan P Böttcher, Marc Beyer, Felix Meissner, Zeinab Abdullah, Jil Sander, Bastian Höchst, Sarah Eickhoff, Jan C Rieckmann, Caroline Russo, Tanja Bauer, Tobias Flecken, Dominik Giesen, Daniel Engel, Steffen Jung, Dirk H Busch, Ulrike Protzer, Robert Thimme, Matthias Mann, Christian Kurts, Joachim L Sc

The role of RIP2 in p38 MAPK activation in the stressed heart.

RIP2 在应激心脏中 p38 MAPK 激活中的作用

Jacquet Sebastien, Nishino Yasuhiro, Kumphune Sarawut, Sicard Pierre, Clark James E, Kobayashi Koichi S, Flavell Richard A, Eickhoff Jan, Cotten Matt, Marber Michael S