日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Trafficking of a nitrogenase FeMo-cofactor assembly intermediate

固氮酶 FeMo 辅因子组装中间体的运输

Schneider, Florian F; Martin Del Campo, Julia S; Zhang, Lin; Dean, Dennis R; Einsle, Oliver

Stabilizing Plasmodium falciparum proteins for small molecule drug discovery

稳定恶性疟原虫蛋白以用于小分子药物发现

Amann, Marius; Sträßer, Tim; Einsle, Oliver; Günther, Stefan

Conformational protection of molybdenum nitrogenase by Shethna protein II

Shethna蛋白II对钼固氮酶的构象保护作用

Franke, Philipp; Freiberger, Simon; Zhang, Lin; Einsle, Oliver

From Pharmacophore to Warhead: NAD(+)-Targeting Triazoles as Mechanism-Based Sirtuin Inhibitors

从药效团到活性位点:靶向 NAD(+) 的三唑类化合物作为基于机制的 Sirtuin 抑制剂

Friedrich, Florian; Meleshin, Marat; Papenkordt, Niklas; Gaitzsch, Lena; Prucker, Isabel; Borso, Marco; Ruprecht, Jan; Vorreiter, Christopher; Rast, Sabrina; Zhang, Lin; Schiedel, Matthias; Sippl, Wolfgang; Imhof, Axel; Jessen, Henning J; Einsle, Oliver; Schutkowski, Mike; Jung, Manfred

Small Protein Domains as Potential Spin Labels for In Vitro, Cellular, and Light-Induced Dipolar EPR Spectroscopy

小蛋白结构域作为体外、细胞和光诱导偶极电子顺磁共振波谱的潜在自旋标记

Günter, Andreas; Ciuti, Susanna; Denkhaus, Lukas; Sappler, Anna; Orian, Laura; Gerhardt, Stefan; Einsle, Oliver; Weber, Stefan; Di Valentin, Marilena; Schleicher, Erik

Efficient Crystallization of Apo Sirt2 for Small-Molecule Soaking and Structural Analysis of Ligand Interactions.

高效结晶 Apo Sirt2 用于小分子浸泡和配体相互作用的结构分析

Friedrich Florian, Schiedel Matthias, Swyter Sören, Zhang Lin, Sippl Wolfgang, Schutkowski Mike, Einsle Oliver, Jung Manfred

Structure-Guided Design of a KMT9 Inhibitor Prodrug with Cellular Activity.

基于结构的KMT9抑制剂前药设计及其细胞活性

Wang Sheng, Barthes Nicolas P F, Urban Sylvia, Hazai Viktor I, Klein Sebastian O, Pappert Tabea, Kümmel Paul, Heller Nicolas, Bacher Johannes, Staudt Maximilian, Ruprecht Jan, Peng Ling, Sum Manuela, Berlin Christopher, Sarraf Daad, Regenass Pierre, Warstat Robin, Walz Johannes, Mishra Pankaj, Zhang Lin, Einsle Oliver, Günther Stefan, Breit Bernhard, Metzger Eric, Jung Manfred, Schüle Roland

Structural evolution of nitrogenase over 3 billion years

固氮酶在30亿年间的结构演化

Cuevas Zuviría, Bruno; Detemple, Franka; Amritkar, Kaustubh; Garcia, Amanda K; Seefeldt, Lance; Einsle, Oliver; Kaçar, Betül

A Novel Inhibitor against the Bromodomain Protein 1 of the Malaria Pathogen Plasmodium Falciparum

一种针对疟原虫(恶性疟原虫)溴结构域蛋白1的新型抑制剂

Amann, Marius; Warstat, Robin; Rechten, Kay Kristin; Theuer, Philip; Schustereder, Magdalena; Clavey, Sophie; Breit, Bernhard; Einsle, Oliver; Hügle, Martin; Petter, Michaela; Günther, Stefan

Escherichia coli Triheme Enzyme YhjA: Structure and Reactivity

大肠杆菌三血红素酶 YhjA:结构和反应性

Hewitt, Patrick; Seidel, Julian; Wüst, Anja; Smith, Meghan; Maiocco, Stephanie J; Shternberg, Stephanie; Hoffmann, Maren; Spatzal, Thomas; Gerhardt, Stefan; Einsle, Oliver; Elliott, Sean J