日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Indole Peptidomimetics Show Potent and Selective Activity against Drug-Resistant Plasmodium falciparum

吲哚肽模拟物对耐药性恶性疟原虫表现出强效且选择性的活性

Januário, Marcelo Augusto Pereira; Valdes, Talita Alvarenga; Maluf, Sarah El Chamy; Mendes, Giovana Rossi; Bonatto, Vinicius; Moura, Igor M R; Mourão, Penina S; Corrêa, Arlene G; Guido, Rafael Victorio Carvalho

Fluorescent Marinoquinoline Derivative as Inhibitors of Plasmodium falciparum: SAR Analysis, Mode of Action and In Vivo Studies

荧光马林喹啉衍生物作为恶性疟原虫抑制剂:构效关系分析、作用机制及体内研究

Santos Barbosa, Patricia; Souza, Guilherme Eduardo; Maluf, Sarah El Chamy; Bonatto, Vinícius; Moura, Caio Silva; Mendes, Giovana Rossi; Valdes, Talita Alvarenga; Annunciato, Yasmin; Rossetto, Barbara Dos Santos; Ventura, Priscilla Dantas de Souza; Ortin, Gilberto Gaspar Duarte; da Silva, Wellington; Icimoto, Marcelo Yudi; Ferreira, Amália Dos Santos; Cruz, Fabio C; Teles, Carolina B G; Pereira, Dhelio B; Cassiano, Gustavo Capatti; Santana, Sofia; Prudêncio, Miguel; Barbosa, Camila S; Moura, Igor M R; Giampauli, Renan Marcel; De Sousa, Irene Layane; Rocco, Silvana Aparecida; Gazarini, Marcos L; Correia, Carlos Roque Duarte; Aguiar, Anna Caroline Campos; Guido, Rafael Victorio Carvalho

Indole-2-carboxamides Optimization for Antiplasmodial Activity

吲哚-2-甲酰胺类化合物的抗疟活性优化

Kumar, Malkeet; Ahmad, Anees; Aguiar, Anna Caroline Campos; Maluf, Sarah El Chamy; Shamim, Anwar; Ferrer, Mariana; Souza, Guilherme E; Gazarini, Marcos L; Pereira, Dhelio B; von Geldern, Thomas W; Baud, Delphine; Jones, Barry; Mondal, Susanta Kumar; Willis, Paul A; Guido, Rafael Victorio Carvalho; Dias, Luiz Carlos

Marine Guanidine Alkaloids Inhibit Malaria Parasites Development in In Vitro, In Vivo and Ex Vivo Assays

海洋胍类生物碱在体外、体内和离体试验中均能抑制疟原虫的发育

Mendes, Giovana Rossi; Noronha, Anderson L; Moura, Igor M R; Moreira, Natália Menezes; Bonatto, Vinícius; Barbosa, Camila S; Maluf, Sarah El Chamy; Souza, Guilherme Eduardo de; de Amorim, Marcelo Rodrigues; Aguiar, Anna Caroline Campos; Cruz, Fabio C; Ferreira, Amália Dos Santos; Teles, Carolina B G; Pereira, Dhelio B; Hajdu, Eduardo; Ferreira, Antonio G; Berlinck, Roberto G S; Guido, Rafael Victorio Carvalho

High-Throughput Analysis of the Flagella FliK-Dependent Surfaceome and Secretome in Bacillus thuringiensis

对苏云金芽孢杆菌鞭毛FliK依赖性表面组和分泌组的高通量分析

Mouawad, Carine; Awad, Mireille Kallassy; Rodrigues-Machado, Carine; Henry, Céline; Sanchis-Borja, Vincent; El Chamy, Laure

Synthesis, Structure−Activity Relationships, and Parasitological Profiling of Brussonol Derivatives as New Plasmodium falciparum Inhibitors

Brussonol 衍生物作为新型恶性疟原虫抑制剂的合成、结构-活性关系和寄生虫学分析

Camila S Barbosa, Anees Ahmad, Sarah El Chamy Maluf, Igor M R Moura, Guilherme E Souza, Giovanna A H Guerra, Roberto R Moraes Barros, Marcos L Gazarini, Anna C C Aguiar, Antonio C B Burtoloso, Rafael V C Guido

A novel anti-dipteran Bacillus thuringiensis strain: Unusual Cry toxin genes in a highly dynamic plasmid environment

一种新型抗双翅目昆虫的苏云金芽孢杆菌菌株:高度动态质粒环境中的异常Cry毒素基因

Fayad, Nancy; Kambris, Zakaria; El Chamy, Laure; Mahillon, Jacques; Kallassy Awad, Mireille

Protein Phosphatase 4 Negatively Regulates the Immune Deficiency-NF-κB Pathway during the Drosophila Immune Response

蛋白磷酸酶 4 在果蝇免疫反应过程中对免疫缺陷-NF-κB 通路起负向调控作用

Layale Salem Wehbe, Dana Barakat, Adrian Acker, Rita El Khoury, Jean-Marc Reichhart, Nicolas Matt, Laure El Chamy

Overexpression of Plasmodium falciparum M1 Aminopeptidase Promotes an Increase in Intracellular Proteolysis and Modifies the Asexual Erythrocytic Cycle Development

恶性疟原虫M1氨肽酶的过表达促进细胞内蛋白水解增加并改变无性红细胞周期发育

Hoff, Carolina C; Azevedo, Mauro F; Thurler, Adriana B; Maluf, Sarah El Chamy; Melo, Pollyana M S; Del Rivero, Maday Alonso; González-Bacerio, Jorge; Carmona, Adriana K; Budu, Alexandre; Gazarini, Marcos L

The fliK Gene Is Required for the Resistance of Bacillus thuringiensis to Antimicrobial Peptides and Virulence in Drosophila melanogaster

fliK基因是苏云金芽孢杆菌对抗菌肽产生抗性以及在果蝇中致病所必需的。

Attieh, Zaynoun; Mouawad, Carine; Rejasse, Agnès; Jehanno, Isabelle; Perchat, Stéphane; Hegna, Ida K; Økstad, Ole A; Kallassy Awad, Mireille; Sanchis-Borja, Vincent; El Chamy, Laure