日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fat or flat? The impact of dipole moment vectors on non-covalent interactions between aromatic tags and macromolecules

胖还是扁?偶极矩矢量对芳香标签与大分子间非共价相互作用的影响

Holub, Josef; Jílková, Adéla; Lemke, Carina; Cianni, Lorenzo; Spiwoková, Petra; Horn, Martin; Breuer, Christian; Leontovyč, Adrian; Brynda, Jiří; Mertlíková-Kaiserová, Helena; Chanová, Marta; Dos Reis Rocho, Fernanda; Montanari, Carlos A; El-Sakkary, Nelly; Caffrey, Conor R; Gütschow, Michael; Hnyk, Drahomír; Mareš, Michael; Fanfrlík, Jindřich

Enhancing schistosomiasis drug discovery approaches with optimized proteasome substrates.

利用优化的蛋白酶体底物增强血吸虫病药物发现方法

Silva Elany B, Jiang Zhenze, Liu Chenxi, Fajtová Pavla, Teixeira Thaiz R, de Castro Fiorini Maia Giovana, Liu Lawrence J, El-Sakkary Nelly, Skinner Danielle E, Syed Ali, Wang Steven C, Caffrey Conor R, O'Donoghue Anthony J

Identification of Substituted 4-Aminocinnolines as Broad-Spectrum Antiparasitic Agents

鉴定取代的4-氨基喹啉类化合物作为广谱抗寄生虫药物

Spaulding, Andrew; Sharma, Amrita; Giardini, Miriam A; Hoffman, Benjamin; Bernatchez, Jean A; McCall, Laura-Isobel; Calvet, Claudia M; Ackermann, Jasmin; Souza, Julia M; Thomas, Diane; Millard, Caroline C; Devine, William G; Singh, Baljinder; Silva, Everton M; Leed, Susan E; Roncal, Norma E; Penn, Erica C; Erath, Jessey; Kumar, Gaurav; Sepulveda, Yadira; Garcia, Arnold; Rodriguez, Ana; El-Sakkary, Nelly; Sciotti, Richard J; Campbell, Robert F; Momper, Jeremiah D; McKerrow, James H; Caffrey, Conor R; Siqueira-Neto, Jair L; Pollastri, Michael P; Mensa-Wilmot, Kojo; Ferrins, Lori

Bioactivity of Farnesyltransferase Inhibitors Against Entamoeba histolytica and Schistosoma mansoni

法尼基转移酶抑制剂对溶组织内阿米巴和曼氏血吸虫的生物活性

Probst, Alexandra; Nguyen, Thi N; El-Sakkary, Nelly; Skinner, Danielle; Suzuki, Brian M; Buckner, Frederick S; Gelb, Michael H; Caffrey, Conor R; Debnath, Anjan

Phenotypic, chemical and functional characterization of cyclic nucleotide phosphodiesterase 4 (PDE4) as a potential anthelmintic drug target.

环核苷酸磷酸二酯酶 4 (PDE4) 作为潜在驱虫药物靶点的表型、化学和功能表征

Long Thavy, Rojo-Arreola Liliana, Shi Da, El-Sakkary Nelly, Jarnagin Kurt, Rock Fernando, Meewan Maliwan, Rascón Alberto A Jr, Lin Lin, Cunningham Katherine A, Lemieux George A, Podust Larissa, Abagyan Ruben, Ashrafi Kaveh, McKerrow James H, Caffrey Conor R

A novel G protein-coupled receptor of Schistosoma mansoni (SmGPR-3) is activated by dopamine and is widely expressed in the nervous system.

曼氏血吸虫的一种新型 G 蛋白偶联受体 (SmGPR-3) 可被多巴胺激活,并在神经系统中广泛表达

El-Shehabi Fouad, Taman Amira, Moali Lorena S, El-Sakkary Nelly, Ribeiro Paula