日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

First-in-Class Dual PDGFR/Carbonic Anhydrase IX/XII Inhibitors: 6,7-Dimethoxyquinoline-Sulfonamides as Promising Antileukemic Agents

首创的双重PDGFR/碳酸酐酶IX/XII抑制剂:6,7-二甲氧基喹啉磺酰胺类药物作为有前景的抗白血病药物

Roshdy, Eslam; Řezníčková, Eva; Elbadawi, Mostafa M; Celik, Ismail; Giovannuzzi, Simone; Veselá, Denisa; Vojáčková, Veronika; Krňávková, Petra; Nocentini, Alessio; Supuran, Claudiu T; Kryštof, Vladimír; Eldehna, Wagdy M; Abe, Manabu

Synthesis and Biological Evaluation of Imidazopyridine-Isatin Hybrids as Inhibitors of Leishmania major Growth

咪唑并吡啶-靛红杂合物作为利什曼原虫生长抑制剂的合成及生物学评价

El Hassab, Mahmoud A; Eldehna, Wagdy M; Elsayed, Zainab M; Elbadawi, Mostafa M; Negmeldin, Ahmed T; Balaha, Marwa; Nasralla, Sherry N; Monir, Rehan; Ibrahim, Tamer M; Abe, Manabu; Tawfik, Haytham O; Bekhit, Adnan A; Hemeda, Loah R

Discovery of potent bisindole-based pyrazolopyridine derivatives as topoisomerase inhibitors: DNA damage induction and synergistic antileukemic activity

发现强效的基于双吲哚的吡唑并吡啶衍生物作为拓扑异构酶抑制剂:DNA损伤诱导和协同抗白血病活性

Eldehna, Wagdy M; Tawfik, Haytham O; Veselá, Denisa; Peřina, Miroslav; Negmeldin, Ahmed T; Elsayed, Zainab M; Majrashi, Taghreed A; Vojáčková, Veronika; Elbadawi, Mostafa M; Shaldam, Moataz A; Kryštof, Vladimír; Abdel-Aziz, Hatem A

Pyrazole-triazole hybrids as kinase-triad inhibitors: a triple-target strategy for synergistic anticancer therapy

吡唑-三唑杂合物作为激酶三联体抑制剂:一种用于协同抗癌治疗的三靶点策略

Elkotamy, Mahmoud S; Elgohary, Mohamed K; Fakhry, Mariam M; Albakri, Mohamed E; Naglah, Abdelrahman A; Almehizia, Abdulrahman A; Naglah, Ahmed M; Fares, Mohamed; Tawfik, Haytham O; Eldehna, Wagdy M; Abdel-Aziz, Hatem A

Synthesis of new trans-ferulic acid derivatives as potential anticancer agents and VEGFR-2 inhibitors

合成新型反式阿魏酸衍生物作为潜在的抗癌剂和VEGFR-2抑制剂

Mohie, Asmaa N; Doheim, Mahmoud A; El Masry, Ragab A; Gomaa, Ayman M; Salem, Rofaida; Tawfik, Haytham O; Eldehna, Wagdy M

Real-world comparative effectiveness of FOLFIRINOX versus gemcitabine/nab-paclitaxel in metastatic pancreatic cancer: prognostic impact of metastatic site and burden in a Middle Eastern cohort

FOLFIRINOX方案与吉西他滨/白蛋白紫杉醇方案治疗转移性胰腺癌的真实世界疗效比较:转移部位和肿瘤负荷对中东人群预后的影响

Eldehna, Wesal M; Elbarbry, Fawzy; Shakra, Rafat Abu; Elrasad, Shaimaa A; Morsi, Zeinab A; Soaida, Shamel M; Wagdy, Wael M; Aljohani, Abrar I; Abbas, Ramy M

Correction: Formulation of zein nanoparticles for augmenting the anti-inflammatory activity of dexketoprofen

更正:制备玉米醇溶蛋白纳米颗粒以增强右酮洛芬的抗炎活性

El Hassab, Mahmoud A; Ibrahim, Mona H; Abdel Mageed, Sherif S; Mahmoud, Abdulla M A; Othman Ahmed, Zainab Sabry; Mosallam, Shaimaa; Abdelbari, Manar Adel; Khaleel, Eman F; El Hasab, Maram A; Elsayyad, Asmaa; Allam, Shady; Eltabeeb, Moaz A; Negmeldin, Ahmed T; Eldehna, Wagdy M; Albash, Rofida

Discovery of Novel Piperidinyl-Based Benzoxazole Derivatives as Anticancer Agents Targeting VEGFR-2 and c-Met Kinases

发现新型哌啶基苯并恶唑衍生物作为靶向VEGFR-2和c-Met激酶的抗癌药物

Eldehna, Wagdy M; Elsayed, Zainab M; Elnagar, Mohamed R; El-Said, Ahmed H; Majrashi, Taghreed A; Negmeldin, Ahmed T; Saleh, Abdulrahman M; Elrayess, Ranza; Elnahriry, Khaled A; Chen, Zhi-Long; Elagawany, Mohamed; Tawfik, Haytham O

Formulation of zein nanoparticles for augmenting the anti-inflammatory activity of dexketoprofen.

制备玉米醇溶蛋白纳米颗粒以增强右酮洛芬的抗炎活性

El Hassab Mahmoud A, Ibrahim Mona H, Abdel Mageed Sherif S, Mahmoud Abdulla M A, Othman Ahmed Zainab Sabry, Mosallam Shaimaa, Abdelbari Manar Adel, Khaleel Eman F, El Hasab Maram A, Elsayyad Asmaa, Allam Shady, Eltabeeb Moaz A, Negmeldin Ahmed T, Eldehna Wagdy M, Albash Rofida

Multi-stage structure-based virtual screening approach combining 3D pharmacophore, docking and molecular dynamic simulation towards the identification of potential selective PARP-1 inhibitors

结合三维药效团、分子对接和分子动力学模拟的多阶段基于结构的虚拟筛选方法,用于鉴定潜在的选择性PARP-1抑制剂

El Hassab, Mahmoud A; Eldehna, Wagdy M; Hassan, Ghaneya S; Abou-Seri, Sahar M