日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: Shoushtari et al. A Phase Ib Study of Sotrastaurin, a PKC Inhibitor, and Alpelisib, a PI3Kα Inhibitor, in Patients with Metastatic Uveal Melanoma. Cancers 2021, 13, 5504

更正:Shoushtari 等人,《Sotrastaurin(一种 PKC 抑制剂)和 Alpelisib(一种 PI3Kα 抑制剂)治疗转移性葡萄膜黑色素瘤患者的 Ib 期研究》,Cancers 2021, 13, 5504

Shoushtari, Alexander N; Khan, Shaheer; Komatsubara, Kimberly; Feun, Lynn; Acquavella, Nicolas; Singh-Kandah, Shahnaz; Negri, Tiffany; Nesson, Alexandra; Abbate, Kelly; Cremers, Serge; Musi, Elgilda; Ambrosini, Grazia; Lee, Shing; Schwartz, Gary K; Carvajal, Richard D

Protein biomarkers for response to XPO1 inhibition in haematologic malignancies

血液系统恶性肿瘤对 XPO1 抑制反应的蛋白质生物标志物

Tulasigeri M Totiger, Sana Chaudhry, Elgilda Musi, Jumana Afaghani, Skye Montoya, Frank Owusu-Ansah, Stanley Lee, Gary Schwartz, Virginia Klimek, Justin Taylor

The GPER Agonist LNS8801 Induces Mitotic Arrest and Apoptosis in Uveal Melanoma Cells

GPER 激动剂 LNS8801 诱导葡萄膜黑色素瘤细胞有丝分裂停滞和凋亡

Grazia Ambrosini, Christopher A Natale, Elgilda Musi, Tina Garyantes, Gary K Schwartz

Transcriptional analysis of metastatic uveal melanoma survival nominates NRP1 as a therapeutic target

转移性葡萄膜黑色素瘤生存的转录分析提名NRP1作为治疗靶点

Riyue Bao, Oliver Surriga, Daniel J Olson, Jacob B Allred, Carrie A Strand, Yuanyuan Zha, Timothy Carll, Brian W Labadie, Bruno R Bastos, Marcus Butler, David Hogg, Elgilda Musi, Grazia Ambrosini, Pamela Munster, Gary K Schwartz, Jason J Luke

A Phase Ib Study of Sotrastaurin, a PKC Inhibitor, and Alpelisib, a PI3Kα Inhibitor, in Patients with Metastatic Uveal Melanoma

PKC 抑制剂 Sotrastaurin 和 PI3Kα 抑制剂 Alpelisib 治疗转移性葡萄膜黑色素瘤患者的 Ib 期研究

Alexander N Shoushtari, Shaheer Khan, Kimberly Komatsubara, Lynn Feun, Nicolas Acquavella, Shahnaz Singh-Kandah, Tiffany Negri, Alexandra Nesson, Kelly Abbate, Serge Cremers, Elgilda Musi, Grazia Ambrosini, Shing Lee, Gary K Schwartz, Richard D Carvajal

Inhibition of NF-κB-Dependent Signaling Enhances Sensitivity and Overcomes Resistance to BET Inhibition in Uveal Melanoma

抑制 NF-κB 依赖性信号可增强葡萄膜黑色素瘤的敏感性并克服对 BET 抑制的抵抗力

Grazia Ambrosini, Catherine Do, Benjamin Tycko, Ronald B Realubit, Charles Karan, Elgilda Musi, Richard D Carvajal, Vivian Chua, Andrew E Aplin, Gary K Schwartz

Preclinical Evaluation of Nintedanib, a Triple Angiokinase Inhibitor, in Soft-tissue Sarcoma: Potential Therapeutic Implication for Synovial Sarcoma

三重血管激酶抑制剂尼达尼布在软组织肉瘤中的临床前评估:对滑膜肉瘤的潜在治疗意义

Parag P Patwardhan, Elgilda Musi, Gary K Schwartz

Significant blockade of multiple receptor tyrosine kinases by MGCD516 (Sitravatinib), a novel small molecule inhibitor, shows potent anti-tumor activity in preclinical models of sarcoma

新型小分子抑制剂 MGCD516(Sitravatinib)可显著阻断多种受体酪氨酸激酶,在肉瘤临床前模型中表现出强大的抗肿瘤活性

Parag P Patwardhan, Kathryn S Ivy, Elgilda Musi, Elisa de Stanchina, Gary K Schwartz

BRD4-targeted therapy induces Myc-independent cytotoxicity in Gnaq/11-mutatant uveal melanoma cells

BRD4 靶向治疗在 Gnaq/11 突变型葡萄膜黑色素瘤细胞中诱导 Myc 独立的细胞毒性

Grazia Ambrosini, Ashley D Sawle, Elgilda Musi, Gary K Schwartz

The phosphoinositide 3-kinase α selective inhibitor BYL719 enhances the effect of the protein kinase C inhibitor AEB071 in GNAQ/GNA11-mutant uveal melanoma cells

磷脂酰肌醇3-激酶α选择性抑制剂BYL719可增强蛋白激酶C抑制剂AEB071在GNAQ/GNA11突变型葡萄膜黑色素瘤细胞中的作用。

Musi, Elgilda; Ambrosini, Grazia; de Stanchina, Elisa; Schwartz, Gary K