日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fragment Merging, Growing, and Linking Identify New Trypanothione Reductase Inhibitors for Leishmaniasis

片段合并、生长和连接可鉴定用于治疗利什曼病的新型锥虫硫酮还原酶抑制剂

Cécile Exertier, Alessandra Salerno, Lorenzo Antonelli, Annarita Fiorillo, Riccardo Ocello, Francesca Seghetti, Jessica Caciolla, Elisa Uliassi, Matteo Masetti, Eleonora Fiorentino, Stefania Orsini, Trentina Di Muccio, Andrea Ilari, Maria Laura Bolognesi

Integrating a quinone substructure into histone deacetylase inhibitors to cope with Alzheimer's disease and cancer

将醌亚结构整合到组蛋白去乙酰化酶抑制剂中以应对阿尔茨海默病和癌症

Melissa Guardigni, Giulia Greco, Eleonora Poeta, Alan Santini, Elisa Tassinari, Christian Bergamini, Chiara Zalambani, Angela De Simone, Vincenza Andrisano, Elisa Uliassi, Barbara Monti, Maria Laura Bolognesi, Carmela Fimognari, Andrea Milelli

Discovery of Sustainable Drugs for Neglected Tropical Diseases: Cashew Nut Shell Liquid (CNSL)-Based Hybrids Target Mitochondrial Function and ATP Production in Trypanosoma brucei

发现可持续的被忽视的热带疾病药物:基于腰果壳液 (CNSL) 的混合物靶向布氏锥虫的线粒体功能和 ATP 产生

Michela Cerone, Elisa Uliassi, Federica Prati, Godwin U Ebiloma, Leandro Lemgruber, Christian Bergamini, David G Watson, Thais de A M Ferreira, Gabriella Simões Heyn Roth Cardoso, Luiz A Soares Romeiro, Harry P de Koning, Maria Laura Bolognesi

Structure-Based Design of 3-(4-Aryl-1H-1,2,3-triazol-1-yl)-Biphenyl Derivatives as P2Y14 Receptor Antagonists

基于结构的设计 3-(4-芳基-1H-1,2,3-三唑-1-基)-联苯衍生物作为 P2Y14 受体拮抗剂

Anna Junker, Ramachandran Balasubramanian, Antonella Ciancetta, Elisa Uliassi, Evgeny Kiselev, Chiara Martiriggiano, Kevin Trujillo, Giorgi Mtchedlidze, Leah Birdwell, Kyle A Brown, T Kendall Harden, Kenneth A Jacobson