日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Linsitinib Decreases Thyrotropin-Induced Thyroid Hormone Synthesis by Inhibiting Crosstalk Between Thyroid-Stimulating Hormone and Insulin-Like Growth Factor 1 Receptors in Human Thyrocytes In Vitro and In Vivo in Mice.

Linsitinib 通过抑制人甲状腺细胞中促甲状腺激素和胰岛素样生长因子 1 受体之间的串扰,降低促甲状腺激素诱导的甲状腺激素合成(体外和体内小鼠)

Boutin Alisa, Eliseeva Elena, Templin Scott, Marcus-Samuels Bernice, Anderson D Eric, Gershengorn Marvin C, Neumann Susanne

Impaired striatal glutathione-ascorbate metabolism induces transient dopamine increase and motor dysfunction.

纹状体谷胱甘肽-抗坏血酸代谢受损会导致短暂的多巴胺增加和运动功能障碍

Malik Mohd Yaseen, Guo Fei, Asif-Malik Aman, Eftychidis Vasileios, Barkas Nikolaos, Eliseeva Elena, Timm Kerstin N, Wolska Aleksandra, Bergin David, Zonta Barbara, Ratz-Wirsching Veronika, von Hörsten Stephan, Walton Mark E, Magill Peter J, Nerlov Claus, Minichiello Liliana

Ablation of TrkB from Enkephalinergic Precursor-Derived Cerebellar Granule Cells Generates Ataxia

从脑啡肽能前体细胞衍生的颗粒细胞中敲除TrkB会导致共济失调

Eliseeva, Elena; Malik, Mohd Yaseen; Minichiello, Liliana

Discovery of a Positive Allosteric Modulator of the Thyrotropin Receptor: Potentiation of Thyrotropin-Mediated Preosteoblast Differentiation In Vitro

发现一种促甲状腺激素受体的正向变构调节剂:体外增强促甲状腺激素介导的前成骨细胞分化

Neumann, Susanne; Eliseeva, Elena; Boutin, Alisa; Barnaeva, Elena; Ferrer, Marc; Southall, Noel; Kim, David; Hu, Xin; Morgan, Sarah J; Marugan, Juan J; Gershengorn, Marvin C

β-Arrestin-1 mediates thyrotropin-enhanced osteoblast differentiation

β-Arrestin-1介导促甲状腺激素增强的成骨细胞分化

Boutin, Alisa; Eliseeva, Elena; Gershengorn, Marvin C; Neumann, Susanne

A selective TSH receptor antagonist inhibits stimulation of thyroid function in female mice

选择性TSH受体拮抗剂可抑制雌性小鼠甲状腺功能的刺激

Neumann, Susanne; Nir, Eshel A; Eliseeva, Elena; Huang, Wenwei; Marugan, Juan; Xiao, Jingbo; Dulcey, Andrés E; Gershengorn, Marvin C

A new small-molecule antagonist inhibits Graves' disease antibody activation of the TSH receptor

一种新型小分子拮抗剂可抑制格雷夫斯病抗体激活促甲状腺激素受体。

Neumann, Susanne; Eliseeva, Elena; McCoy, Joshua G; Napolitano, Giorgio; Giuliani, Cesidio; Monaco, Fabrizio; Huang, Wenwei; Gershengorn, Marvin C

The Synthesis and Evaluation of Dihydroquinazolin-4-ones and Quinazolin-4-ones as Thyroid Stimulating Hormone Receptor Agonists

二氢喹唑啉-4-酮和喹唑啉-4-酮作为促甲状腺激素受体激动剂的合成与评价

Englund, Erika E; Neumann, Susanne; Eliseeva, Elena; McCoy, Joshua G; Titus, Steven; Zheng, Wei; Southall, Noel; Shin, Paul; Leister, William; Thomas, Craig J; Inglese, James; Austin, Christopher P; Gershengorn, Marvin C; Huang, Wenwei

A small molecule inverse agonist for the human thyroid-stimulating hormone receptor

人促甲状腺激素受体的小分子反向激动剂

Neumann, Susanne; Huang, Wenwei; Eliseeva, Elena; Titus, Steve; Thomas, Craig J; Gershengorn, Marvin C