日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Critical Assessment of a Structure-Based Pipeline for Targeting the Long Noncoding RNA MALAT1

对靶向长链非编码RNA MALAT1的结构导向型流程的关键评估

Aguti, Riccardo; Bernetti, Mattia; Elisi, Gian Marco; Cavalli, Andrea; Masetti, Matteo

Small molecules targeting the eubacterial β-sliding clamp discovered by combined in silico and in vitro screening approaches

通过结合计算机模拟和体外筛选方法,发现了靶向真细菌β-滑动钳的小分子。

Alessia Caputo ,Gian Marco Elisi ,Elisabetta Levati ,Giulia Barotti ,Sara Sartini ,Jerome Wagner ,Dominique Y Burnouf ,Simone Ottonello ,Silvia Rivara ,Barbara Montanini

Identification of a Quinone Derivative as a YAP/TEAD Activity Modulator from a Repurposing Library

从化合物重定位库中鉴定出一种醌衍生物作为YAP/TEAD活性调节剂。

Lauriola, Angela; Uliassi, Elisa; Santucci, Matteo; Bolognesi, Maria Laura; Mor, Marco; Scalvini, Laura; Elisi, Gian Marco; Gozzi, Gaia; Tagliazucchi, Lorenzo; Marverti, Gaetano; Ferrari, Stefania; Losi, Lorena; D'Arca, Domenico; Costi, Maria Paola

Free-Energy Simulations Support a Lipophilic Binding Route for Melatonin Receptors

自由能模拟支持褪黑激素受体的亲脂性结合途径

Elisi, Gian Marco; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Rivara, Silvia

An Optimized Workflow for the Discovery of New Antimicrobial Compounds Targeting Bacterial RNA Polymerase Complex Formation

针对细菌 RNA 聚合酶复合物形成的新型抗菌化合物的优化工作流程

Alessia Caputo, Sara Sartini, Elisabetta Levati, Ilaria Minato, Gian Marco Elisi, Adriana Di Stasi, Catherine Guillou, Peter G Goekjian, Pierre Garcia, David Gueyrard, Stéphane Bach, Arnaud Comte, Simone Ottonello, Silvia Rivara, Barbara Montanini

New classes of potent heparanase inhibitors from ligand-based virtual screening

基于配体虚拟筛选的新型强效肝素酶抑制剂

Pala, Daniele; Scalvini, Laura; Elisi, Gian Marco; Lodola, Alessio; Mor, Marco; Spadoni, Gilberto; Ferrara, Fabiana F; Pavoni, Emiliano; Roscilli, Giuseppe; Milazzo, Ferdinando M; Battistuzzi, Gianfranco; Rivara, Silvia; Giannini, Giuseppe