A Structure-based Design Approach for Generating High Affinity BRD4 D1-Selective Chemical Probes
基于结构的设计方法,用于生成高亲和力 BRD4 D1 选择性化学探针
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c01779
Huarui Cui, Anand Divakaran, Zachariah J Hoell, Mikael O Ellingson, Cole R Scholtz, Huda Zahid, Jorden A Johnson, Elizabeth C Griffith, Clifford T Gee, Amani L Lee, Shalil Khanal, Ke Shi, Hideki Aihara, Vijay H Shah, Richard E Lee, Daniel A Harki, William C K Pomerantz