日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Amino acid and viral binding by the high-affinity Cationic Amino acid Transporter 1 (CAT1) from Mus musculus

小鼠高亲和力阳离子氨基酸转运蛋白1 (CAT1) 对氨基酸和病毒的结合

Ye, Mingda; Liang, Zhu; Zhou, Daming; Pike, Ashley C W; Wang, SiYi; Wang, Dong; Bakshi, Souvika; Brooke, Laurent; Williams, Eleanor P; Elkins, Jonathan M; Kessler, Benedikt M; Stuart, David I; Sauer, David B

Tetrahydropyrazolopyridinones as a Novel Class of Potent and Highly Selective LIMK Inhibitors

四氢吡唑并吡啶酮类化合物作为一类新型高效高选择性LIMK抑制剂

Baldwin, Alex G; Foley, David W; Jones, D Heulyn; Lee, Hyunah; Collins, Ross; Wahab, Ben; Pedder, Josephine H; Waters, Loren; Paine, Marie; Schino, Lauramariú; Feng, Gui Jie; Kariuki, Benson M; Elkins, Jonathan M; Atack, John R; Ward, Simon E

Discovery of MDI-114215: A Potent and Selective LIMK Inhibitor To Treat Fragile X Syndrome.

MDI-114215 的发现:一种强效且选择性的 LIMK 抑制剂,可用于治疗脆性 X 综合征

Baldwin Alex G, Foley David W, Collins Ross, Lee Hyunah, Jones D Heulyn, Wahab Ben, Waters Loren, Pedder Josephine, Paine Marie, Feng Gui Jie, Privitera Lucia, Ashall-Kelly Alexander, Thomas Carys, Gillespie Jason A, Schino Lauramariú, Belelli Delia, Rocha Cecilia, Maussion Gilles, Krahn Andrea I, Durcan Thomas M, Elkins Jonathan M, Lambert Jeremy J, Atack John R, Ward Simon E

Toward target 2035: EUbOPEN - a public-private partnership to enable & unlock biology in the open

迈向2035年目标:EUbOPEN——一项旨在促进和开放生物学的公私合作项目

Tredup, Claudia; Ackloo, Suzanne; Beck, Hartmut; Brown, Peter J; Bullock, Alex N; Ciulli, Alessio; Dikic, Ivan; Edfeldt, Kristina; Edwards, Aled M; Elkins, Jonathan M; Farin, Henner F; Fon, Edward A; Gstaiger, Matthias; Günther, Judith; Gustavsson, Anna-Lena; Häberle, Sandra; Isigkeit, Laura; Huber, Kilian V M; Kotschy, Andras; Krämer, Oliver; Leach, Andrew R; Marsden, Brian D; Matsui, Hisanori; Merk, Daniel; Montel, Florian; Mulder, Monique P C; Müller, Susanne; Owen, Dafydd R; Proschak, Ewgenij; Röhm, Sandra; Stolz, Alexandra; Sundström, Michael; von Delft, Frank; Willson, Timothy M; Arrowsmith, Cheryl H; Knapp, Stefan

Updated protein domain annotation of the PARP protein family sheds new light on biological function

PARP蛋白家族蛋白质结构域注释的更新为生物学功能提供了新的见解

Suskiewicz, Marcin J; Munnur, Deeksha; Strømland, Øyvind; Yang, Ji-Chun; Easton, Laura E; Chatrin, Chatrin; Zhu, Kang; Baretić, Domagoj; Goffinont, Stéphane; Schuller, Marion; Wu, Wing-Fung; Elkins, Jonathan M; Ahel, Dragana; Sanyal, Sumana; Neuhaus, David; Ahel, Ivan

SGC-AAK1-1: A Chemical Probe Targeting AAK1 and BMP2K

SGC-AAK1-1:一种靶向AAK1和BMP2K的化学探针

Wells, Carrow; Couñago, Rafael M; Limas, Juanita C; Almeida, Tuanny L; Cook, Jeanette Gowen; Drewry, David H; Elkins, Jonathan M; Gileadi, Opher; Kapadia, Nirav R; Lorente-Macias, Alvaro; Pickett, Julie E; Riemen, Alexander; Ruela-de-Sousa, Roberta R; Willson, Timothy M; Zhang, Cunyu; Zuercher, William J; Zutshi, Reena; Axtman, Alison D

Development of 2-(4-pyridyl)-benzimidazoles as PKN2 chemical tools to probe cancer

开发2-(4-吡啶基)-苯并咪唑类化合物作为PKN2化学工具用于癌症研究

Scott, Fiona; Fala, Angela M; Pennicott, Lewis E; Reuillon, Tristan D; Massirer, Katlin B; Elkins, Jonathan M; Ward, Simon E

Solution structures and biophysical analysis of full-length group A PAKs reveal they are monomeric and auto-inhibited in cis

全长A组PAK的溶液结构和生物物理分析表明,它们是单体,并且在顺式作用下发生自身抑制。

Sorrell, Fiona J; Kilian, Lena Marie; Elkins, Jonathan M

Development of Pyridine-based Inhibitors for the Human Vaccinia-related Kinases 1 and 2

开发用于抑制人痘苗病毒相关激酶 1 和 2 的吡啶类抑制剂

Serafim, Ricardo A M; de Souza Gama, Fernando H; Dutra, Luiz A; Dos Reis, Caio V; Vasconcelos, Stanley N S; da Silva Santiago, André; Takarada, Jéssica E; Di Pillo, Fúlvia; Azevedo, Hatylas; Mascarello, Alessandra; Elkins, Jonathan M; Massirer, Katlin B; Gileadi, Opher; Guimarães, Cristiano R W; Couñago, Rafael M

Crystal structure of human RIOK2 bound to a specific inhibitor

人RIOK2与特异性抑制剂结合的晶体结构

Wang, Jing; Varin, Thibault; Vieth, Michal; Elkins, Jonathan M