Second-Generation AURKA-Targeting PROTACs: Structural Optimization toward in Vivo Degradation in Neuroblastoma
第二代靶向AURKA的PROTAC:针对神经母细胞瘤体内降解的结构优化
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c01271
Krols, Simon; Rishfi, Muhammad; Martens, Fien; Van Hauwermeiren, Anouk; Sanders, Ellen; De Sutter, Pieter-Jan; Vermeulen, An; De Wever, Kaat; Bekaert, Sarah-Lee; Dolman, M Emmy M; Tax, Gabor; Kamili, Alvin; Fletcher, Jamie I; Depestel, Lisa; De Wilde, Bram; Durinck, Kaat; Van Calenbergh, Serge