日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Modulating food intake by nasal application of peptides targeting melanocortin 4 receptor and ghrelin receptor systems

通过鼻腔施用靶向黑皮质素4受体和胃饥饿素受体系统的肽来调节食物摄入量

Özbay, Benginur; Jülke, Eva-Maria; List, Moritz; Nowicki, Marcin; Els-Heindl, Sylvia; Immig, Kerstin; Mörl, Karin; Bechmann, Ingo; Beck-Sickinger, Annette G

Photoinduced receptor confinement drives ligand-independent GPCR signaling

光诱导受体限制驱动配体独立的GPCR信号传导

M Florencia Sánchez, Sylvia Els-Heindl, Annette G Beck-Sickinger, Ralph Wieneke, Robert Tampé

Cyclic Derivatives of the Chemerin C-Terminus as Metabolically Stable Agonists at the Chemokine-like Receptor 1 for Cancer Treatment

趋化因子C端环状衍生物作为趋化因子样受体1的代谢稳定激动剂用于癌症治疗

Fischer, Tobias F; Czerniak, Anne S; Weiß, Tina; Zellmann, Tristan; Zielke, Lina; Els-Heindl, Sylvia; Beck-Sickinger, Annette G

Tryptophan Analogues with Fixed Side-Chain Orientation: Expanding the Scope

具有固定侧链取向的色氨酸类似物:拓展研究范围

Nicke, Lennart; Horx, Philip; Müller, Ronny; Els-Heindl, Sylvia; Geyer, Armin

Development of a ghrelin receptor inverse agonist for positron emission tomography

用于正电子发射断层扫描的生长素释放肽受体反向激动剂的开发

Ralf Bergmann, Constance Chollet, Sylvia Els-Heindl, Martin Ullrich, Nicole Berndt, Jens Pietzsch, Domokos Máthé, Michael Bachmann, Annette G Beck-Sickinger

Structural Model of Ghrelin Bound to its G Protein-Coupled Receptor.

生长素释放肽与其 G 蛋白偶联受体结合的结构模型

Bender Brian Joseph, Vortmeier Gerrit, Ernicke Stefan, Bosse Mathias, Kaiser Anette, Els-Heindl Sylvia, Krug Ulrike, Beck-Sickinger Annette, Meiler Jens, Huster Daniel

Side Chain Orientation of Tryptophan Analogues Determines Agonism and Inverse Agonism in Short Ghrelin Peptides

色氨酸类似物的侧链取向决定了短链生长素释放肽的激动剂和反向激动剂作用

Nicke, Lennart; Müller, Ronny; Geyer, Armin; Els-Heindl, Sylvia

Development of Fluorinated Non-Peptidic Ghrelin Receptor Ligands for Potential Use in Molecular Imaging

开发用于分子成像的氟化非肽类生长素释放肽受体配体

Moldovan, Rareş-Petru; Els-Heindl, Sylvia; Worm, Dennis J; Kniess, Torsten; Kluge, Michael; Beck-Sickinger, Annette G; Deuther-Conrad, Winnie; Krügel, Ute; Brust, Peter

Expression, Functional Characterization, and Solid-State NMR Investigation of the G Protein-Coupled GHS Receptor in Bilayer Membranes

双层膜中G蛋白偶联GHS受体的表达、功能表征和固态核磁共振研究

Schrottke, Stefanie; Kaiser, Anette; Vortmeier, Gerrit; Els-Heindl, Sylvia; Worm, Dennis; Bosse, Mathias; Schmidt, Peter; Scheidt, Holger A; Beck-Sickinger, Annette G; Huster, Daniel

Peptide mini-scaffold facilitates JNK3 activation in cells

肽微型支架促进细胞内JNK3的激活

Zhan, Xuanzhi; Stoy, Henriette; Kaoud, Tamer S; Perry, Nicole A; Chen, Qiuyan; Perez, Alejandro; Els-Heindl, Sylvia; Slagis, Jack V; Iverson, Tina M; Beck-Sickinger, Annette G; Gurevich, Eugenia V; Dalby, Kevin N; Gurevich, Vsevolod V