Optimization of a Novel Quinazolinone-Based Series of Transient Receptor Potential A1 (TRPA1) Antagonists Demonstrating Potent in Vivo Activity
优化一系列新型基于喹唑啉酮的瞬时受体电位 A1 (TRPA1) 拮抗剂,展示出强效的体内活性
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.6b00039
Laurie B Schenkel, Philip R Olivieri, Alessandro A Boezio, Holly L Deak, Renee Emkey, Russell F Graceffa, Hakan Gunaydin, Angel Guzman-Perez, Josie H Lee, Yohannes Teffera, Weiya Wang, Beth D Youngblood, Violeta L Yu, Maosheng Zhang, Narender R Gavva, Sonya G Lehto, Stephanie Geuns-Meyer